SCHEMBL2554892

SCHEMBL2554892

CNC(=O)NC(=O)C(C)Oc1ccccc1C=O

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.67
ALDH1A1 P00352 6/20 0.43
GAA P10253 2/20 0.43
ACHE P22303 1/20 0.42
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
SMN1; SMN2 Q16637 4/20 0.39
HPGD P15428 2/20 0.39
HTT P42858 1/20 0.39
ATM Q13315 1/20 0.39
SRC P12931 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
KMT2A Q03164 2/20 0.38
TSHR P16473 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
RECQL P46063 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15331058 0.88 LMNA (0.50) LMNAALDH1A1GAAACHEADRA2A
SCHEMBL2554388 0.85 SMN1; SMN2 (0.56) LMNAALDH1A1GAAADRA2AADRA2B
SCHEMBL2557678 0.84 LMNA (0.47) LMNAALDH1A1GAAACHEADRA2A
SCHEMBL2553758 0.82 LMNA (0.51) LMNAALDH1A1GAASMN1; SMN2HPGD
SCHEMBL2562943 0.81 ALDH1A1 (0.46) LMNAALDH1A1GAAADRA2AADRA2B
SCHEMBL15330283 0.79 LMNA (0.57) LMNAALDH1A1GAASMN1; SMN2HPGD
SCHEMBL29952275 0.79 SMN1; SMN2 (0.52) LMNAALDH1A1GAAADRA2AADRA2B
SCHEMBL29952101 0.79 ALDH1A1 (0.43) LMNAALDH1A1GAAADRA2AADRA2B
SCHEMBL15058014 0.78 KMT2A (0.46) LMNAALDH1A1GAAACHEADRA2A
SCHEMBL15331066 0.78 PTGDR2 (0.43) LMNAALDH1A1GAAADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-11225655-B2 Bi-functional complexes and methods for making and using such complexes NUEVOLUTION A/S (DK) 2022-01-18 US disclosed
EP-3540059-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2019-09-18 EP disclosed
EP-2558577-B1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION AS (DK) 2018-12-12 EP disclosed
US-20130281324-A1 BI-FUNCTINAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2013-10-24 US disclosed
EP-2558577-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2013-02-20 EP disclosed
WO-2011127933-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2011-10-20 WO disclosed