SCHEMBL2555729

SCHEMBL2555729

COC(=O)Cc1ccccc1-c1cccnc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 3/20 0.51
ALDH1A1 P00352 4/20 0.49
KDM4E B2RXH2 1/20 0.49
NPC1 O15118 1/20 0.49
MAPK1 P28482 1/20 0.49
ADORA2A P29274 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2D6 P10635 2/20 0.45
CYP2C19 P33261 2/20 0.45
HSD17B10 Q99714 2/20 0.45
CLK4 Q9HAZ1 2/20 0.45
USP2 O75604 1/20 0.45
ALOX15 P16050 1/20 0.45
EPHX1 P07099 1/20 0.45
PTGS2 P35354 1/20 0.44
KCNH2 Q12809 1/20 0.44
CYP11B1 P15538 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2557632 0.85 EPHX1 (0.43) KCNA5ALDH1A1KDM4EMEN1KMT2A
SCHEMBL7353766 0.84 KMT2A (0.51) KDM4EKMT2ACYP2D6
Hydrogen Sulfide SCHEMBL28029150 0.83 KMT2A (0.50) KDM4EKMT2ACYP2D6
SCHEMBL6237509 0.83 FFAR1 (0.51) ALDH1A1KDM4ENPC1MAPK1KCNH2
SCHEMBL3735688 0.81 KCNA5 (0.59) KCNA5ALDH1A1KDM4EKMT2ACYP1A2
SCHEMBL2175358 0.80 KCNA5 (0.54) KCNA5ALDH1A1KMT2ACYP1A2CYP3A4
SCHEMBL28321278 0.80 ACLY (0.48) ALDH1A1NPC1MEN1KMT2A
SCHEMBL9285273 0.79 KCNA5 (0.59) KCNA5ALDH1A1KMT2ACYP1A2CYP3A4
SCHEMBL5956551 0.79 NR4A2 (0.45) ALDH1A1KDM4ENPC1MAPK1MEN1
SCHEMBL14810463 0.78 SLC2A1 (0.48) ALDH1A1KDM4ENPC1MAPK1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011123937-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2011-10-13 WO disclosed
WO-2011123937-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2011-10-13 WO disclosed