SCHEMBL2555843

SCHEMBL2555843

CC(C(=O)Nc1ccc2[nH]ncc2c1)c1ccccc1

nearest known ligand 0.73

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 9/20 0.64
ROCK1 Q13464 9/20 0.64
NPC1 O15118 5/20 0.63
RAB9A P51151 4/20 0.63
JAK2 O60674 3/20 0.63
ALDH1A1 P00352 2/20 0.56
MAPT P10636 2/20 0.56
HPGD P15428 1/20 0.56
ALOX12 P18054 1/20 0.56
JAK1 P23458 2/20 0.55
TMIGD3 P0DMS9 1/20 0.53
ADORA1 P30542 1/20 0.53
KDM4E B2RXH2 1/20 0.53
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2555842 1.00 ROCK2 (0.64) ROCK2ROCK1NPC1RAB9AJAK2
SCHEMBL20661258 0.86 ROCK2 (0.59) ROCK2ROCK1NPC1RAB9AJAK2
SCHEMBL14863508 0.85 ROCK2 (0.62) ROCK2ROCK1NPC1RAB9AJAK2
SCHEMBL20661185 0.85 ROCK2 (0.62) ROCK2ROCK1NPC1RAB9AJAK2
SCHEMBL14863507 0.85 ROCK2 (0.62) ROCK2ROCK1NPC1RAB9AJAK2
SCHEMBL23429984 0.85 ROCK2 (0.64) ROCK2ROCK1NPC1RAB9AJAK2
SCHEMBL19699462 0.84 ROCK2 (0.71) ROCK2ROCK1NPC1RAB9AJAK2
SCHEMBL23429978 0.83 ROCK2 (0.62) ROCK2ROCK1NPC1RAB9AJAK2
SCHEMBL20661259 0.82 ROCK2 (0.58) ROCK2ROCK1NPC1RAB9AJAK2
SCHEMBL20661200 0.82 ROCK2 (0.59) ROCK2ROCK1NPC1RAB9AJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011123937-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2011-10-13 WO disclosed