SCHEMBL2555879

SCHEMBL2555879

CC(C(=O)O)N(C)c1ccccc1C1Nc2ccc(C(=O)O)cc2CC1(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
ALDH1A1 P00352 2/20 0.36
POLB P06746 2/20 0.36
GAA P10253 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
APOBEC3A P31941 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
MAPT P10636 2/20 0.32
KDM4E B2RXH2 1/20 0.32
MASP2 O00187 1/20 0.31
HSPA1A P0DMV8 1/20 0.31
CD44 P16070 1/20 0.31
PTPN1 P18031 1/20 0.31
MSN P26038 1/20 0.31
CDC25B P30305 1/20 0.31
AKT1 P31749 1/20 0.31
PTPN7 P35236 1/20 0.31
EZH2 Q15910 1/20 0.31
SRD5A2 P31213 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2534264 0.80 DYRK2 (0.41) MEN1KMT2AALDH1A1POLBGAA
SCHEMBL15495131 0.78 ALDH1A1 (0.35) MEN1KMT2AALDH1A1POLBGAA
SCHEMBL2530126 0.78 ALDH1A1 (0.40) MEN1KMT2AALDH1A1POLBGAA
SCHEMBL2532897 0.76 GCK (0.38) MEN1KMT2AALDH1A1GAAMAPT
SCHEMBL2533782 0.75 NEU3 (0.38) MEN1KMT2AALDH1A1POLBGAA
SCHEMBL12219890 0.75 KMO (0.43) MEN1KMT2AALDH1A1POLBGAA
SCHEMBL2535888 0.74 SIRT2 (0.34) MEN1KMT2AALDH1A1POLBGAA
SCHEMBL2529037 0.74 ALDH1A1 (0.32) MEN1KMT2AALDH1A1POLBGAA
SCHEMBL2574768 0.74 MAPT (0.40) MEN1KMT2AALDH1A1GAAL3MBTL1
SCHEMBL2532334 0.73 KDM4E (0.41) MEN1KMT2AALDH1A1POLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2558449-A1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2013-02-20 EP disclosed
WO-2011128251-A1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2011-10-20 WO disclosed