SCHEMBL255607

SCHEMBL255607

CCOc1cnc(-c2cccc(Cc3nn(-c4cccc(N)c4)ccc3=O)c2)nc1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35
MET P08581 9/20 0.34
CSNK1D P48730 1/20 0.34
DHFR P00374 1/20 0.34
FGFR3 P22607 1/20 0.33
KDR P35968 1/20 0.33
PDE10A Q9Y233 1/20 0.33
HSD17B13 Q7Z5P4 1/20 0.33
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
GRM2 Q14416 1/20 0.32
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12518001 0.89 MET (0.45) METPDE10APPARGPPARA
SCHEMBL12516728 0.89 TTK (0.39) METFGFR3KDRHSD17B13PPARG
SCHEMBL13274725 0.89 MET (0.34) METFGFR3KDRHSD17B13PPARG
SCHEMBL256018 0.89 TP53 (0.35) TP53CYP3A4METCSNK1DDHFR
SCHEMBL2222009 0.89 MET (0.43) TP53METCSNK1DFGFR3KDR
SCHEMBL12516348 0.88 MET (0.36) METDHFRFGFR3KDRHSD17B13
SCHEMBL13274895 0.86 MET (0.44) MET
SCHEMBL13274873 0.86 MET (0.43) METFGFR3KDRHSD17B13
SCHEMBL2221788 0.85 MET (0.34) METFGFR3KDRHSD17B13
SCHEMBL2224454 0.85 FYN (0.38) CYP3A4METFGFR3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012030633-A1 TYROSINE KINASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-03-08 WO disclosed