SCHEMBL256018

SCHEMBL256018

CCOc1cnc(-c2cccc(Cc3nn(-c4cccc(N)c4)ccc3=S)c2)nc1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35
DHFR P00374 1/20 0.34
MET P08581 8/20 0.33
CSNK1D P48730 1/20 0.33
FGFR3 P22607 1/20 0.31
KDR P35968 1/20 0.31
NOTUM Q6P988 2/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
PKM P14618 1/20 0.31
KMT2A Q03164 1/20 0.31
MERTK Q12866 1/20 0.31
PPARG P37231 1/20 0.31
PPARA Q07869 1/20 0.31
NQO2 P16083 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL255607 0.89 TP53 (0.35) TP53CYP3A4DHFRMETCSNK1D
SCHEMBL163957 0.86 MET (0.43) METNQO2
SCHEMBL173429 0.84 BRD4 (0.34) METPPARGPPARANQO2
SCHEMBL12516728 0.80 TTK (0.39) METFGFR3KDRMEN1NPC1
SCHEMBL12518001 0.79 MET (0.45) METPPARGPPARA
SCHEMBL2222009 0.78 MET (0.43) TP53METCSNK1DFGFR3KDR
SCHEMBL13274725 0.78 MET (0.34) METFGFR3KDRNPC1PPARG
SCHEMBL12516348 0.77 MET (0.36) DHFRMETFGFR3KDR
SCHEMBL2224454 0.76 FYN (0.38) CYP3A4METFGFR3KDRNPC1
SCHEMBL164341 0.76 MET (0.38) METFGFR3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012030633-A1 TYROSINE KINASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-03-08 WO disclosed