SCHEMBL2556372

SCHEMBL2556372

CNC(=O)NC(=O)CN1CCCC(C=O)C1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.49
ALDH1A1 P00352 3/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.41
KDM4E B2RXH2 3/20 0.36
HPGD P15428 1/20 0.36
SIGMAR1 Q99720 3/20 0.34
CHRM5 P08912 2/20 0.34
CHRM1 P11229 2/20 0.34
KMT2A Q03164 2/20 0.34
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM3 P20309 1/20 0.34
BCHE P06276 1/20 0.34
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2558206 0.88 L3MBTL1 (0.41) L3MBTL1ALDH1A1MAPK1KDM4EHPGD
SCHEMBL2557592 0.85 L3MBTL1 (0.61) L3MBTL1ALDH1A1MAPK1SMN1; SMN2KDM4E
SCHEMBL2560295 0.84 L3MBTL1 (0.45) L3MBTL1ALDH1A1MAPK1SMN1; SMN2KDM4E
SCHEMBL2571616 0.83 L3MBTL1 (0.43) L3MBTL1ALDH1A1MAPK1SMN1; SMN2KDM4E
SCHEMBL2555995 0.83 L3MBTL1 (0.44) L3MBTL1ALDH1A1MAPK1SMN1; SMN2KDM4E
SCHEMBL2555959 0.83 L3MBTL1 (0.42) L3MBTL1ALDH1A1MAPK1SMN1; SMN2KDM4E
SCHEMBL2556697 0.82 ALDH1A1 (0.44) L3MBTL1ALDH1A1MAPK1SMN1; SMN2KDM4E
SCHEMBL2557667 0.81 ALDH1A1 (0.49) L3MBTL1ALDH1A1MAPK1SMN1; SMN2KDM4E
SCHEMBL2556555 0.80 KDM4E (0.46) L3MBTL1ALDH1A1MAPK1SMN1; SMN2KDM4E
SCHEMBL2558609 0.80 CHRM5 (0.49) L3MBTL1ALDH1A1SMN1; SMN2KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-11225655-B2 Bi-functional complexes and methods for making and using such complexes NUEVOLUTION A/S (DK) 2022-01-18 US disclosed
EP-3540059-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2019-09-18 EP disclosed
EP-2558577-B1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION AS (DK) 2018-12-12 EP disclosed
US-20130281324-A1 BI-FUNCTINAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2013-10-24 US disclosed
EP-2558577-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2013-02-20 EP disclosed
WO-2011127933-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2011-10-20 WO disclosed