SCHEMBL25565710

SCHEMBL25565710

C=C1CCC(N2C(=O)c3cccc(CC(C)C)c3C2=O)C(=O)N1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 19/20 0.55
CRBN Q96SW2 19/20 0.55
IKZF3 Q9UKT9 2/20 0.52
TNF P01375 1/20 0.52
IL1B P01584 1/20 0.52
TBXA2R P21731 1/20 0.52
IKZF1 Q13422 1/20 0.52
ALDH1A1 P00352 1/20 0.48
CHRM2 P08172 1/20 0.48
OPRM1 P35372 1/20 0.48
CYP1A2 P05177 1/20 0.48
TSHR P16473 1/20 0.48
TDP1 Q9NUW8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23589806 0.89 DDB1 (0.69) DDB1CRBNIKZF3TNFIL1B
SCHEMBL18878464 0.84 DDB1 (0.56) DDB1CRBNIKZF3TNFIL1B
SCHEMBL25467701 0.84 DDB1 (0.56) DDB1CRBNIKZF3TNFIL1B
SCHEMBL25467690 0.84 DDB1 (0.56) DDB1CRBNIKZF3TNFIL1B
SCHEMBL23707575 0.82 DDB1 (0.77) DDB1CRBNIKZF3TNFIL1B
SCHEMBL25876249 0.81 DDB1 (0.55) DDB1CRBNIKZF3TNFIL1B
SCHEMBL15502840 0.81 DDB1 (0.58) DDB1CRBNIKZF3TNFIL1B
SCHEMBL20317527 0.81 DDB1 (0.80) DDB1CRBNIKZF3TNFIL1B
SCHEMBL677366 0.81 CRBN (0.77) DDB1CRBNIKZF3TNFIL1B
SCHEMBL17246852 0.81 CRBN (0.77) DDB1CRBNIKZF3TNFIL1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240025863-A1 SOS1 PROTEIN DEGRADERS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND THEIR THERAPEUTIC APPLICATIONS BIOTHERYX, INC. 2024-01-25 US disclosed
US-20230293702-A1 QUINAZOLINES, PHARMACEUTICAL COMPOSITIONS, AND THERAPEUTIC APPLICATIONS BIOTHERYX, INC. 2023-09-21 US disclosed
US-20230158157-A1 POTENT AND SELECTIVE DEGRADERS OF ALK DANA-FARBER CANCER INSTITUTE, INC. (US) 2023-05-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230293702-A1 QUINAZOLINES, PHARMACEUTICAL COMPOSITIONS, AND THERAPEUTIC APPLICATIONS RAB1A, SOS1, IQGAP1 DDB1 2095/4885CRBN 3656/4885IKZF3 3769/4885
US-20230158157-A1 POTENT AND SELECTIVE DEGRADERS OF ALK ALK, ERBB2, PDGFRB DDB1 1650/4885CRBN 500/4885IKZF3 2131/4885
US-20240025863-A1 SOS1 PROTEIN DEGRADERS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND THEIR THERAPEUTIC APPLICATIONS SOS1, SOS2, SOST DDB1 985/4885CRBN 474/4885IKZF3 2458/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.