SCHEMBL255722

SCHEMBL255722

Nc1cccc(Cc2nn(-c3cccc(N)c3)ccc2=O)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
MAPT P10636 1/20 0.38
POLB P06746 1/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
ABHD6 Q9BV23 2/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP2C9 P11712 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
MAOA P21397 2/20 0.35
MAOB P27338 2/20 0.35
MGLL Q99685 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2223282 0.93 CYP2C9 (0.43) PARP1MEN1KMT2APOLBCYP11B1
SCHEMBL13274755 0.88 GRM5 (0.44) PARP1CYP11B1CYP11B2CYP19A1
SCHEMBL13275009 0.88 PARP1 (0.37) PARP1MAPTPOLBCYP11B1CYP11B2
SCHEMBL13275315 0.87 PARP1 (0.39) PARP1MEN1KMT2ACYP11B1CYP11B2
SCHEMBL13275429 0.86 PARP1 (0.38) PARP1MEN1KMT2ACYP11B1CYP11B2
SCHEMBL13274914 0.84 PARP1 (0.37) PARP1MAPTCYP11B1CYP11B2ABHD6
SCHEMBL173258 0.83 PARP1 (0.38) PARP1MEN1KMT2AABHD6ALDH1A1
SCHEMBL13275207 0.83 CCNB2 (0.38) PARP1MAPTPOLBCYP11B1CYP11B2
SCHEMBL255607 0.81 TP53 (0.35)
SCHEMBL12518001 0.78 MET (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012030633-A1 TYROSINE KINASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-03-08 WO disclosed