SCHEMBL25575759

SCHEMBL25575759

CCOc1ccc(C)cc1N1CCC(=O)NC1=O

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 9/20 0.49
DDB1 Q16531 8/20 0.49
MEN1 O00255 4/20 0.45
KMT2A Q03164 4/20 0.45
TSHR P16473 2/20 0.45
POLB P06746 1/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
L3MBTL1 Q9Y468 3/20 0.41
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23065973 0.85 DDB1 (0.52) CRBNDDB1MEN1KMT2ATSHR
SCHEMBL25905759 0.84 ALDH1A1 (0.47) CRBNDDB1MEN1KMT2ATSHR
SCHEMBL21408861 0.83 TSHR (0.48) CRBNDDB1MEN1KMT2ATSHR
SCHEMBL30148827 0.83 TSHR (0.48) CRBNDDB1MEN1KMT2ATSHR
SCHEMBL25575719 0.82 CRBN (0.60) CRBNDDB1ALDH1A1GAA
SCHEMBL25575744 0.81 CRBN (0.48) CRBNDDB1MEN1KMT2AKDM4E
SCHEMBL25122532 0.79 CRBN (0.67) CRBNDDB1MEN1KMT2ATSHR
SCHEMBL25596152 0.77 DDB1 (0.41) CRBNDDB1MEN1KMT2APOLB
SCHEMBL25074350 0.76 CRBN (0.55) CRBNDDB1MEN1KMT2AKDM4E
SCHEMBL31607794 0.76 CRBN (0.55) CRBNDDB1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4393922-A1 IRAK4 DEGRADATION AGENT, AND PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Leadingtac Pharmaceutical Co. Ltd. (CN) 2024-07-03 EP disclosed
EP-4328219-A1 SOS1 DEGRADING AGENT AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF Shanghai Leadingtac Pharmaceutical Co. Ltd. (CN) 2024-02-28 EP disclosed
EP-4194457-A1 COMPOUND FOR TARGETING AND DEGRADING PROTEIN, AND PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Leadingtac Pharmaceutical Co., Ltd. (CN) 2023-06-14 EP disclosed