SCHEMBL2558686

SCHEMBL2558686

O=Cc1cccc(-c2ccnc(C(=O)O)c2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRIM24 O15164 1/20 0.59
TRIM33 Q9UPN9 1/20 0.59
KMO O15229 4/20 0.51
UNG P13051 1/20 0.50
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 3/20 0.47
KDM6B O15054 1/20 0.47
TET3 O43151 1/20 0.47
KDM4A O75164 1/20 0.47
BBOX1 O75936 1/20 0.47
MAPT P10636 1/20 0.47
KDM5A P29375 1/20 0.47
KDM5C P41229 1/20 0.47
ASPH Q12797 1/20 0.47
KDM4D Q6B0I6 1/20 0.47
TET2 Q6N021 1/20 0.47
ALKBH5 Q6P6C2 1/20 0.47
KDM7A Q6ZMT4 1/20 0.47
KDM8 Q8N371 1/20 0.47
TET1 Q8NFU7 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2563186 0.83 KMO (0.58) TRIM24TRIM33KMOKDM4EALDH1A1
SCHEMBL8922592 0.83 KDM4E (0.57) TRIM24TRIM33KMOUNGKDM4E
SCHEMBL2558804 0.81 TRIM24 (0.60) TRIM24TRIM33KMOUNGKDM4E
SCHEMBL725162 0.81 KMO (0.62) KMOKDM4EALDH1A1KDM6BTET3
SCHEMBL30800092 0.80 KMO (0.71) KMOKDM4EALDH1A1KDM6BTET3
SCHEMBL7513922 0.80 KMO (0.71) KMOKDM4EALDH1A1KDM6BTET3
SCHEMBL29068408 0.80 KDM4E (0.53) TRIM24TRIM33KMOUNGKDM4E
SCHEMBL3642765 0.78 KMO (0.56) KMOKDM4EALDH1A1KDM6BTET3
SCHEMBL15329552 0.77 UNG (0.63) TRIM24TRIM33KMOUNGKDM4E
SCHEMBL23201148 0.77 KMO (0.65) KMOKDM4EALDH1A1KDM6BTET3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-11225655-B2 Bi-functional complexes and methods for making and using such complexes NUEVOLUTION A/S (DK) 2022-01-18 US disclosed
EP-3540059-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2019-09-18 EP disclosed
EP-2558577-B1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION AS (DK) 2018-12-12 EP disclosed
US-20130281324-A1 BI-FUNCTINAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2013-10-24 US disclosed
EP-2558577-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2013-02-20 EP disclosed
WO-2011127933-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2011-10-20 WO disclosed