SCHEMBL2558718

SCHEMBL2558718

O=Cc1cccn1-c1ccc(C(=O)O)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.68
POLB P06746 8/20 0.64
APEX1 P27695 5/20 0.64
RECQL P46063 5/20 0.64
TDP1 Q9NUW8 5/20 0.64
L3MBTL1 Q9Y468 5/20 0.64
HTT P42858 1/20 0.64
PTP4A3 O75365 1/20 0.58
ALDH1A1 P00352 7/20 0.57
FHIT P49789 1/20 0.56
DNMT1 P26358 3/20 0.54
MCL1 Q07820 3/20 0.54
NSD2 O96028 2/20 0.54
EP300 Q09472 1/20 0.51
KAT8 Q9H7Z6 1/20 0.51
MAPT P10636 3/20 0.49
NR4A1 P22736 2/20 0.49
MAPK1 P28482 1/20 0.49
PTPN7 P35236 1/20 0.49
HSD17B10 Q99714 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15330143 0.82 POLB (0.72) ATMPOLBAPEX1RECQLTDP1
SCHEMBL1127259 0.81 ATM (1.00) ATMPOLBAPEX1RECQLTDP1
SCHEMBL25240419 0.80 ATM (0.69) ATMPOLBAPEX1RECQLTDP1
SCHEMBL9042897 0.77 ALDH1A1 (0.62) ATMTDP1L3MBTL1HTTALDH1A1
SCHEMBL28775954 0.77 ATM (0.69) ATMPOLBAPEX1RECQLTDP1
SCHEMBL1419333 0.77 ATM (0.69) ATMPOLBRECQLTDP1L3MBTL1
SCHEMBL6634976 0.77 ATM (0.69) ATMPOLBAPEX1RECQLTDP1
SCHEMBL6052462 0.77 ATM (0.69) ATMPOLBL3MBTL1HTTALDH1A1
SCHEMBL3211700 0.77 ATM (0.69) ATMPOLBRECQLTDP1L3MBTL1
SCHEMBL2562622 0.75 PTPN7 (0.51) ATMPOLBAPEX1RECQLTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3634907-B1 MODIFIED NANOSTRUCTURED CARBON MATRIX, CONTAINING SUCH A MATRIX SYSTEM AND INCLUDING SUCH SYSTEM BIOSENSOR AND A METHOD FOR THE DETERMINATION OF AN ANALYTE IN A SAMPLE USING SUCH BIOSENSOR SYSTEM AS WELL AS THE APPLICATION OF A PYRROLE BENZOIC ACID DERIVATIVE FOR THE MODIFICATION OF THE NANOSTRUCTURED CARBON MATRIX UNIV WARSZAWSKI (PL) 2021-09-08 EP claimed
EP-3634907-A1 MODIFIED NANOSTRUCTURED CARBON MATRIX, CONTAINING SUCH A MATRIX SYSTEM AND INCLUDING SUCH SYSTEM BIOSENSOR AND A METHOD FOR THE DETERMINATION OF AN ANALYTE IN A SAMPLE USING SUCH BIOSENSOR SYSTEM AS WELL AS THE APPLICATION OF A PYRROLE BENZOIC ACID DERIVATIVE FOR THE MODIFICATION OF THE NANOSTRUCTURED CARBON MATRIX Uniwersytet Warszawski (PL) 2020-04-15 EP claimed
WO-2018224980-A1 MODIFIED NANOSTRUCTURED CARBON MATRIX, CONTAINING SUCH A MATRIX SYSTEM AND INCLUDING SUCH SYSTEM BIOSENSOR AND A METHOD FOR THE DETERMINATION OF AN ANALYTE IN A SAMPLE USING SUCH BIOSENSOR SYSTEM AS WELL AS THE APPLICATION OF A PYRROLE BENZOIC ACID DERIVATIVE FOR THE MODIFICATION OF THE NANOSTRUCTURED CARBON MATRIX UNIWERSYTET WARSZAWSKI (PL) 2018-12-13 WO claimed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-11225655-B2 Bi-functional complexes and methods for making and using such complexes NUEVOLUTION A/S (DK) 2022-01-18 US disclosed
EP-3634907-B1 MODIFIED NANOSTRUCTURED CARBON MATRIX, CONTAINING SUCH A MATRIX SYSTEM AND INCLUDING SUCH SYSTEM BIOSENSOR AND A METHOD FOR THE DETERMINATION OF AN ANALYTE IN A SAMPLE USING SUCH BIOSENSOR SYSTEM AS WELL AS THE APPLICATION OF A PYRROLE BENZOIC ACID DERIVATIVE FOR THE MODIFICATION OF THE NANOSTRUCTURED CARBON MATRIX UNIV WARSZAWSKI (PL) 2021-09-08 EP disclosed
EP-3634907-A1 MODIFIED NANOSTRUCTURED CARBON MATRIX, CONTAINING SUCH A MATRIX SYSTEM AND INCLUDING SUCH SYSTEM BIOSENSOR AND A METHOD FOR THE DETERMINATION OF AN ANALYTE IN A SAMPLE USING SUCH BIOSENSOR SYSTEM AS WELL AS THE APPLICATION OF A PYRROLE BENZOIC ACID DERIVATIVE FOR THE MODIFICATION OF THE NANOSTRUCTURED CARBON MATRIX Uniwersytet Warszawski (PL) 2020-04-15 EP disclosed
EP-3540059-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2019-09-18 EP disclosed
WO-2018224980-A1 MODIFIED NANOSTRUCTURED CARBON MATRIX, CONTAINING SUCH A MATRIX SYSTEM AND INCLUDING SUCH SYSTEM BIOSENSOR AND A METHOD FOR THE DETERMINATION OF AN ANALYTE IN A SAMPLE USING SUCH BIOSENSOR SYSTEM AS WELL AS THE APPLICATION OF A PYRROLE BENZOIC ACID DERIVATIVE FOR THE MODIFICATION OF THE NANOSTRUCTURED CARBON MATRIX UNIWERSYTET WARSZAWSKI (PL) 2018-12-13 WO disclosed
EP-2558577-B1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION AS (DK) 2018-12-12 EP disclosed
US-20130281324-A1 BI-FUNCTINAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2013-10-24 US disclosed
EP-2558577-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2013-02-20 EP disclosed
WO-2011127933-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2011-10-20 WO disclosed
WO-2007071840-A2 COMPOUNDS BASED ON FOUR AROMATIC RINGS, PREPARATION AND USES THEREOF CEREP (FR) 2007-06-28 WO disclosed
EP-1327631-A2 Fused heterocyclic compounds, their production and use as angiotensin II antagonists Takeda Chemical Industries, Ltd. (JP) 2003-07-16 EP disclosed
EP-0518033-B1 Fused heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-07-02 EP disclosed
US-5389641-A Fused heterocyclic compounds, having angiotensin II antagonistic activity TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-02-14 US disclosed
EP-0518033-A1 Fused heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-12-16 EP disclosed