SCHEMBL2559262

SCHEMBL2559262

O=CC=C(Cl)c1ccc(Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.46
CES1 P23141 3/20 0.46
TSHR P16473 2/20 0.44
MAPK1 P28482 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
ALOX15 P16050 1/20 0.44
CYP3A4 P08684 1/20 0.44
ATM Q13315 1/20 0.44
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
HSD17B10 Q99714 1/20 0.41
GSK3B P49841 2/20 0.40
SRD5A2 P31213 1/20 0.40
LMNA P02545 3/20 0.39
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP1A2 P05177 1/20 0.37
HPGD P15428 1/20 0.37
ALOX12 P18054 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8338715 1.00 CES2 (0.46) CES2CES1TSHRMAPK1L3MBTL1
SCHEMBL2559260 1.00 CES2 (0.46) CES2CES1TSHRMAPK1L3MBTL1
SCHEMBL17074011 0.80 CES2 (0.44) CES2CES1CA1CA2ALDH1A1
SCHEMBL6708832 0.80 ALDH1A1 (0.45) CES2CES1ATMGSK3BSRD5A2
SCHEMBL2559234 0.80 CES2 (0.44) CES2CES1MAPK1CA1CA2
SCHEMBL23275556 0.80 TPMT (0.43) CA1CA2GSK3B
SCHEMBL23285683 0.80 TPMT (0.43) CA1CA2GSK3B
SCHEMBL12489982 0.80 CES2 (0.44) CES2CES1CA1CA2ALDH1A1
SCHEMBL2559233 0.80 CES2 (0.44) CES2CES1MAPK1CA1CA2
SCHEMBL2559511 0.80 CES2 (0.44) CES2CES1MAPK1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0323625-B1 Process for preparing 3-[2-chloro-2(4-chlorophenyl)-vinyl]-2,2-dimethyl-cyclopropane carboxylic acid BAYER AG (DE) 1992-09-09 EP claimed
US-4897505-A Process for the preparation of 3-(2-chloro-2-(4-chloro-phenyl)-vinyl)-2,2-dimethylcyclopropanecarboxylic acid BAYER AKTIENGESELLSCHAFT (DE) 1990-01-30 US claimed
EP-0323625-A2 Process for preparing 3-[2-chloro-2(4-chlorophenyl)-vinyl]-2,2-dimethyl-cyclopropane carboxylic acid BAYER AG (DE) 1989-07-12 EP claimed
JP-1203350-A None JP disclosed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-11225655-B2 Bi-functional complexes and methods for making and using such complexes NUEVOLUTION A/S (DK) 2022-01-18 US disclosed
EP-3540059-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2019-09-18 EP disclosed
EP-2558577-B1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION AS (DK) 2018-12-12 EP disclosed
US-20130281324-A1 BI-FUNCTINAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2013-10-24 US disclosed
EP-2558577-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2013-02-20 EP disclosed
WO-2011127933-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2011-10-20 WO disclosed
US-4992577-A Preparation of 3-vinyl-substituted 2,2-dimethylcyclopropane-1-carboxylic acids and esters and intermediates therefor BAYER AKTIENGESELLSCHAFT (DE) 1991-02-12 US disclosed
US-4897505-A Process for the preparation of 3-(2-chloro-2-(4-chloro-phenyl)-vinyl)-2,2-dimethylcyclopropanecarboxylic acid BAYER AKTIENGESELLSCHAFT (DE) 1990-01-30 US disclosed
US-4897505-A Process for the preparation of 3-(2-chloro-2-(4-chloro-phenyl)-vinyl)-2,2-dimethylcyclopropanecarboxylic acid BAYER AKTIENGESELLSCHAFT (DE) 1990-01-30 US disclosed
JP-H01203350-A PREPARATION OF 3-(2-CHLORO-2-(4-CHLOROPHENYL)-VINYL)-2,2-DIMETHYLCYCLOPROPANECARBOXYLIC ACID BAYER AG 1989-08-16 JP disclosed
EP-0323625-A2 Process for preparing 3-[2-chloro-2(4-chlorophenyl)-vinyl]-2,2-dimethyl-cyclopropane carboxylic acid BAYER AG (DE) 1989-07-12 EP disclosed
EP-0323625-A2 Process for preparing 3-[2-chloro-2(4-chlorophenyl)-vinyl]-2,2-dimethyl-cyclopropane carboxylic acid BAYER AG (DE) 1989-07-12 EP disclosed
EP-0095047-B1 PROCESS FOR THE PREPARATION OF 3-VINYL-SUBSTITUTED 2,2-DIMETHYL-CYCLOPROPANE-1-CARBOXYLIC ACIDS OR THEIR ESTERS, AND INTERMEDIATE PRODUCTS THEREFOR BAYER AG (DE) 1985-11-27 EP disclosed
EP-0095047-A1 Process for the preparation of 3-vinyl-substituted 2,2-dimethyl-cyclopropane-1-carboxylic acids or their esters, and intermediate products therefor BAYER AG (DE) 1983-11-30 EP disclosed
EP-0019089-A1 5-Aryl-3-(1'-halogen-1'-methyl)ethyl-pent-4-en-carboxylic acid esters, process for their preparation, and their use for the preparation of 3-(2-arylvinyl)-2,2-dimethyl-cyclopropane-1-carboxylic acid esters BAYER AG (DE) 1980-11-26 EP disclosed