SCHEMBL255982

SCHEMBL255982

CCCC(=O)c1cc(N)n(Cc2ccccc2F)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.44
CYP2C19 P33261 2/20 0.44
P2RY14 Q15391 1/20 0.44
ALDH1A1 P00352 5/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
ADORA3 P0DMS8 1/20 0.38
KCNH2 Q12809 1/20 0.38
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
NOD2 Q9HC29 1/20 0.38
CYP2C9 P11712 1/20 0.38
SLC16A3 O15427 1/20 0.37
SLC16A1 P53985 1/20 0.37
MCTS1 Q9ULC4 1/20 0.37
TP53 P04637 1/20 0.37
PKM P14618 5/20 0.37
PKLR P30613 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17611691 0.83 P2RY14 (0.57) CYP1A2CYP2C19P2RY14ALDH1A1KMT2A
SCHEMBL175092 0.82 TP53 (0.47) CYP1A2CYP2C19P2RY14ALDH1A1KMT2A
SCHEMBL30223258 0.82 TP53 (0.47) CYP1A2CYP2C19P2RY14ALDH1A1KMT2A
SCHEMBL14998053 0.81 ALDH1A1 (0.55) CYP1A2CYP2C19P2RY14ALDH1A1KMT2A
SCHEMBL18496413 0.79 TP53 (0.45) CYP1A2CYP2C19P2RY14ALDH1A1KMT2A
SCHEMBL20433971 0.79 ALDH1A1 (0.43) CYP1A2CYP2C19P2RY14ALDH1A1KMT2A
SCHEMBL18672320 0.79 P2RY14 (0.45) CYP1A2CYP2C19P2RY14ALDH1A1KMT2A
SCHEMBL18405007 0.75 CYP1A2 (0.40) CYP1A2CYP2C19P2RY14ALDH1A1KMT2A
SCHEMBL6068367 0.73 TP53 (0.43) CYP1A2P2RY14ALDH1A1KMT2AMEN1
SCHEMBL5766056 0.73 KMT2A (0.46) CYP1A2CYP2C19P2RY14ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012028645-A1 METHOD FOR THE PRODUCTION OF 5-FLUORO-1H-PYRAZOLO[3,4-B]PYRIDINE-3-CARBONITRILE BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-03-08 WO disclosed