SCHEMBL25599287

SCHEMBL25599287

CNc1cccc2c1CN(C(=O)c1c(O)cc(O)c(C)c1OCC1CCCCC1)C2

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRAP1 Q12931 4/20 0.35
HSP90B1 P14625 2/20 0.35
NAMPT P43490 2/20 0.35
SIRT2 Q8IXJ6 1/20 0.34
HSP90AA1 P07900 4/20 0.34
THRA P10827 2/20 0.33
THRB P10828 2/20 0.33
GRM5 P41594 1/20 0.33
ADAM17 P78536 1/20 0.33
SPR P35270 1/20 0.32
HSP90AB1 P08238 2/20 0.32
FABP4 P15090 1/20 0.32
CXCR5 P32302 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31281765 1.00 TRAP1 (0.35) TRAP1HSP90B1NAMPTSIRT2HSP90AA1
SCHEMBL31282001 0.95 TRAP1 (0.36) TRAP1HSP90B1HSP90AA1SPRHSP90AB1
SCHEMBL25599277 0.91 HSP90AA1 (0.39) TRAP1HSP90B1NAMPTSIRT2HSP90AA1
SCHEMBL25250614 0.88 NAMPT (0.34) TRAP1HSP90B1NAMPTSIRT2HSP90AA1
SCHEMBL25254449 0.88 NAMPT (0.35) TRAP1HSP90B1NAMPTSIRT2HSP90AA1
SCHEMBL30377316 0.88 NAMPT (0.35) TRAP1HSP90B1NAMPTSIRT2HSP90AA1
SCHEMBL30377606 0.88 NAMPT (0.34) TRAP1HSP90B1NAMPTSIRT2HSP90AA1
SCHEMBL30377635 0.88 NAMPT (0.33) TRAP1HSP90B1NAMPTSIRT2HSP90AA1
SCHEMBL25254673 0.88 NAMPT (0.33) TRAP1HSP90B1NAMPTSIRT2HSP90AA1
SCHEMBL25210256 0.88 TRAP1 (0.36) TRAP1HSP90B1NAMPTHSP90AA1THRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023094834-A1 ISOINDOLINES AS PMS2 INHIBITORS Neophore Limited (GB) 2023-06-01 WO disclosed