SCHEMBL25599412

SCHEMBL25599412

C=CC(=O)Nc1cc2nc(N3CCCC(OC)C3)n(C)c2cc1C

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSC P53634 11/20 0.40
UCHL3 P15374 1/20 0.40
CTSL P07711 2/20 0.39
CTSB P07858 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
CCNA2 P20248 4/20 0.39
CDK2 P24941 4/20 0.39
CDK7 P50613 4/20 0.39
CCNH P51946 4/20 0.39
MNAT1 P51948 4/20 0.39
CCNT1 O60563 2/20 0.39
CDK9 P50750 2/20 0.39
ACACB O00763 1/20 0.37
CCNK O75909 2/20 0.36
CDK12 Q9NYV4 2/20 0.36
BCL2A1 Q16548 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25681380 1.00 CTSC (0.40) CTSCUCHL3CTSLCTSBCYP1A2
SCHEMBL25682250 0.87 CTSC (0.47) CTSCUCHL3CTSLCTSBCYP1A2
SCHEMBL25599169 0.87 CTSC (0.47) CTSCUCHL3CTSLCTSBCYP1A2
SCHEMBL25682448 0.87 CCNA2 (0.39) CTSCUCHL3CTSLCTSBCYP1A2
SCHEMBL25599216 0.87 CCNA2 (0.39) CTSCUCHL3CTSLCTSBCYP1A2
SCHEMBL25682533 0.87 CCNA2 (0.39) CTSCUCHL3CTSLCTSBCYP1A2
SCHEMBL25599226 0.85 BTK (0.43) CTSCUCHL3CTSLCTSBCYP1A2
SCHEMBL25599985 0.81 CTSC (0.41) CTSCUCHL3CTSLCTSBCYP1A2
SCHEMBL25599228 0.81 UCHL3 (0.40) CTSCUCHL3CTSLCTSBCYP1A2
SCHEMBL25221957 0.77 CCNK (0.48) CCNA2CDK2CDK7CCNHMNAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023102184-A1 BICYCLIC AMINE COMPOUNDS AS CDK12 INHIBITORS INCYTE CORPORATION (US) 2023-06-08 WO disclosed