SCHEMBL2560002

SCHEMBL2560002

O=Cc1c(-c2cc(F)cc(F)c2)nn(-c2ccccc2F)c1Cl

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36
KCNN4 O15554 2/20 0.35
MDM4 O15151 1/20 0.33
MDM2 Q00987 1/20 0.33
MAPK11 Q15759 1/20 0.33
MAPK14 Q16539 1/20 0.33
P2RX7 Q99572 1/20 0.32
PIM1 P11309 1/20 0.32
PIM3 Q86V86 1/20 0.32
PIM2 Q9P1W9 1/20 0.32
GAA P10253 1/20 0.32
ATM Q13315 1/20 0.32
RIPK1 Q13546 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15331264 0.90 PTGER1 (0.35) HPGDKMT2AKCNN4P2RX7
SCHEMBL2556623 0.88 POLB (0.41) HPGDKMT2AKCNN4MAPK14
SCHEMBL15331113 0.88 HPGD (0.39) HPGDKMT2AKCNN4SMN1; SMN2
SCHEMBL2556378 0.86 HPGD (0.36) HPGDKMT2AKCNN4MDM4MDM2
SCHEMBL15330615 0.86 GAA (0.39) HPGDKMT2AKCNN4GAARIPK1
SCHEMBL2558355 0.85 MAPT (0.38) HPGDKMT2AKCNN4MDM4MDM2
SCHEMBL2553185 0.85 KCNN4 (0.35) HPGDKMT2AKCNN4MAPK11MAPK14
SCHEMBL2557971 0.84 SMN1; SMN2 (0.40) GAASMN1; SMN2
SCHEMBL29950987 0.83 KCNN4 (0.42) HPGDKMT2AKCNN4PIM1PIM3
SCHEMBL15329895 0.83 KMT2A (0.39) HPGDKMT2AKCNN4MDM4MDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-11225655-B2 Bi-functional complexes and methods for making and using such complexes NUEVOLUTION A/S (DK) 2022-01-18 US disclosed
EP-3540059-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2019-09-18 EP disclosed
EP-2558577-B1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION AS (DK) 2018-12-12 EP disclosed
US-20130281324-A1 BI-FUNCTINAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2013-10-24 US disclosed
EP-2558577-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2013-02-20 EP disclosed
WO-2011127933-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2011-10-20 WO disclosed