SCHEMBL25604196

SCHEMBL25604196

CC(=O)c1ccc2c(c1O)CN(C(=O)OC(C)(C)C)CC2

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.58
NR1H2 P55055 2/20 0.54
MAPK1 P28482 1/20 0.43
ADORA1 P30542 1/20 0.40
MAPT P10636 3/20 0.40
KDM4E B2RXH2 1/20 0.40
GPR119 Q8TDV5 1/20 0.39
PRMT5 O14744 2/20 0.39
WDR77 Q9BQA1 2/20 0.39
ACACB O00763 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
DRD2 P14416 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
SCN9A Q15858 1/20 0.38
NAMPT P43490 1/20 0.38
DDB1 Q16531 1/20 0.38
CRBN Q96SW2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25604351 0.91 ESR2 (0.53) ESR2NR1H2MAPK1ADORA1MAPT
SCHEMBL25604259 0.90 ESR2 (0.58) ESR2NR1H2MAPK1ADORA1MAPT
SCHEMBL25825899 0.88 ESR2 (0.49) ESR2NR1H2MAPK1GPR119ACACB
SCHEMBL14895889 0.84 ESR2 (0.53) ESR2NR1H2MAPK1MAPTPRMT5
SCHEMBL25604195 0.80 ESR2 (0.54) ESR2MAPK1MAPTDRD2HDAC6
SCHEMBL29097964 0.79 ESR2 (0.63) ESR2NR1H2MAPK1ADORA1MAPT
SCHEMBL30199545 0.79 ESR2 (0.63) ESR2NR1H2MAPK1ADORA1MAPT
SCHEMBL15503203 0.78 ESR2 (0.56) ESR2NR1H2MAPK1ADORA1MAPT
SCHEMBL3693657 0.78 ESR2 (0.59) ESR2NR1H2MAPK1ADORA1MAPT
SCHEMBL30199091 0.78 ESR2 (0.59) ESR2NR1H2MAPK1ADORA1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125944-A1 COMPOUND CONTAINING HETEROCYCLIC RING 正大天晴药业集团股份有限公司 2023-07-06 WO disclosed
WO-2023088406-A1 FUSED IMIDE DERIVATIVE 正大天晴药业集团股份有限公司 2023-05-25 WO disclosed