SCHEMBL25604259

SCHEMBL25604259

CC(=O)c1ccc2c(c1O)CCN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.58
NR1H2 P55055 2/20 0.54
MAPK1 P28482 1/20 0.45
ACACB O00763 1/20 0.44
SCN9A Q15858 1/20 0.43
UCHL1 P09936 1/20 0.43
ADORA1 P30542 2/20 0.43
MAPT P10636 3/20 0.42
KDM4E B2RXH2 1/20 0.42
DDB1 Q16531 2/20 0.40
CRBN Q96SW2 2/20 0.40
NAMPT P43490 1/20 0.40
PARP1 P09874 1/20 0.39
TNKS2 Q9H2K2 1/20 0.39
PARP2 Q9UGN5 1/20 0.39
HDAC1 Q13547 1/20 0.39
GPR119 Q8TDV5 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25604351 0.91 ESR2 (0.53) ESR2NR1H2MAPK1ADORA1MAPT
SCHEMBL25604196 0.90 ESR2 (0.58) ESR2NR1H2MAPK1ACACBSCN9A
SCHEMBL25825899 0.88 ESR2 (0.49) ESR2NR1H2MAPK1ACACBSCN9A
SCHEMBL15503203 0.88 ESR2 (0.56) ESR2NR1H2MAPK1ACACBSCN9A
SCHEMBL17583907 0.86 ESR2 (0.62) ESR2NR1H2MAPK1ACACBSCN9A
SCHEMBL30150249 0.84 ESR2 (0.57) ESR2NR1H2MAPK1ACACBSCN9A
SCHEMBL16039921 0.82 ESR2 (0.58) ESR2NR1H2MAPK1ACACBSCN9A
SCHEMBL31680222 0.80 ESR2 (0.61) ESR2NR1H2MAPK1ACACBSCN9A
SCHEMBL2117366 0.80 ESR2 (0.61) ESR2NR1H2MAPK1ACACBSCN9A
SCHEMBL25604257 0.80 ESR2 (0.54) ESR2MAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125944-A1 COMPOUND CONTAINING HETEROCYCLIC RING 正大天晴药业集团股份有限公司 2023-07-06 WO disclosed
WO-2023088406-A1 FUSED IMIDE DERIVATIVE 正大天晴药业集团股份有限公司 2023-05-25 WO disclosed