SCHEMBL256053

SCHEMBL256053

CC/C=C/c1ccc(N(C)C)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 5/20 0.59
RELA Q04206 1/20 0.57
MAPT P10636 6/20 0.55
MEN1 O00255 4/20 0.55
KMT2A Q03164 4/20 0.55
CASP1 P29466 2/20 0.55
HBB P68871 2/20 0.55
GAA P10253 1/20 0.55
BRCA1 P38398 1/20 0.55
CASP7 P55210 1/20 0.55
SMN1; SMN2 Q16637 4/20 0.53
ALOX15 P16050 2/20 0.53
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
HSD17B3 P37058 1/20 0.52
KDM4E B2RXH2 1/20 0.52
ALDH1A1 P00352 4/20 0.50
LMNA P02545 2/20 0.50
HTT P42858 2/20 0.50
PTGS1 P23219 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL213343 1.00 APP (0.59) APPRELAMAPTMEN1KMT2A
SCHEMBL27870189 0.86 APP (0.70) APPRELAMAPTMEN1KMT2A
SCHEMBL25000571 0.83 APP (0.55) APPRELAMAPTMEN1KMT2A
SCHEMBL1714449 0.81 RELA (0.81) APPRELAMAPTMEN1KMT2A
SCHEMBL13467434 0.81 RELA (0.81) APPRELAMAPTMEN1KMT2A
SCHEMBL7915381 0.81 RELA (0.81) APPRELAMAPTMEN1KMT2A
SCHEMBL1714446 0.81 RELA (0.81) APPRELAMAPTMEN1KMT2A
SCHEMBL3025040 0.81 RELA (0.81) APPRELAMAPTMEN1KMT2A
SCHEMBL10846378 0.81 APP (0.57) APPRELAMAPTMEN1KMT2A
SCHEMBL14329676 0.81 ALDH1A1 (0.61) MAPTMEN1KMT2ACASP1HBB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020112846-A1 SMALL MOLECULE MODULATORS OF SIGMA-1 AND SIGMA-2 RECEPTORS AND USES THEREOF NORTHWESTERN UNIVERSITY (US) 2020-06-04 WO disclosed
EP-2651374-B1 PROCESS FOR DYEING KERATIN FIBRES USING A DIRECT DYE BEARING A DISULFIDE/THIOL/PROTECTED THIOL FUNCTION AND WATER VAPOUR L'ORÉAL (FR) 2018-02-28 EP disclosed
WO-2012028578-A1 SUBSTITUTED FUSED PYRIMIDINONES AND DIHYDROPYRIMIDINONES BAYER CROPSCIENCE AG (DE) 2012-03-08 WO disclosed