SCHEMBL25614993

SCHEMBL25614993

O=c1cccnn1-c1cncc(Br)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
USP8 P40818 1/20 0.39
CHRNB2 P17787 7/20 0.36
CHRNA4 P43681 7/20 0.36
HRH3 Q9Y5N1 4/20 0.36
KCNH2 Q12809 1/20 0.36
ALOX15 P16050 1/20 0.35
HTT P42858 1/20 0.35
EP300 Q09472 1/20 0.34
KAT2B Q92831 1/20 0.34
CHRNB4 P30926 5/20 0.34
CHRNA3 P32297 5/20 0.34
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29151050 0.80 CA12 (0.47) CA12CA1CA2CA9HRH3
SCHEMBL30745148 0.80 CA12 (0.47) CA12CA1CA2CA9HRH3
SCHEMBL29151066 0.78 CA1 (0.60) CA12CA1CA2CA9USP8
SCHEMBL14955293 0.78 CA12 (0.51) CA12CA1CA2CA9HTT
SCHEMBL25614983 0.77 CA12 (0.42) CA12CA1CA2CA9CHRNB2
SCHEMBL14909303 0.73 HTT (0.40) CA12CA1CA2CA9USP8
SCHEMBL15105004 0.73 CA12 (0.59) CA12CA1CA2CA9HRH3
SCHEMBL25614994 0.73 CA12 (0.39) CA12CA1CA2CA9HRH3
SCHEMBL2411328 0.72 CA12 (0.50) CA12CA1CA2CA9USP8
SCHEMBL3043828 0.71 CA12 (0.61) CA12CA1CA2CA9HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023104209-A1 METTL3 INHIBITOR COMPOUND 上海昂阔医药有限公司 2023-06-15 WO disclosed