SCHEMBL25614994

SCHEMBL25614994

C[Si](C)(C)C#Cc1cncc(-n2ncccc2=O)c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
HRH3 Q9Y5N1 4/20 0.35
KCNH2 Q12809 1/20 0.34
GABRA1 P14867 2/20 0.33
GABRG2 P18507 2/20 0.33
GABRB3 P28472 2/20 0.33
GABRA5 P31644 2/20 0.33
GABRA3 P34903 2/20 0.33
GABRA2 P47869 2/20 0.33
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
GRM5 P41594 3/20 0.32
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25614983 0.81 CA12 (0.42) CA12CA1CA2CA9HRH3
SCHEMBL25614740 0.78 GABRA1 (0.37) CA12CA1CA2CA9GABRA1
SCHEMBL25614598 0.75 KDM4E (0.40) GRM5
SCHEMBL25614466 0.74 GRM5 (0.31) GRM5
SCHEMBL25614993 0.73 CA12 (0.45) CA12CA1CA2CA9HRH3
SCHEMBL30811694 0.71 GRM5 (0.31) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL14955293 0.70 CA12 (0.51) CA12CA1CA2CA9CYP3A4
SCHEMBL30811822 0.70 CHRNB2 (0.37) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL22531723 0.69 GRM5 (0.38) GRM5
SCHEMBL29176201 0.68 CYP1A2 (0.30) CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023104209-A1 METTL3 INHIBITOR COMPOUND 上海昂阔医药有限公司 2023-06-15 WO disclosed