SCHEMBL2561567

SCHEMBL2561567

CN(C)c1ccccc1C(=O)n1nc(-c2cccnc2)cc1N

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK3 P07288 6/20 0.56
F2 P00734 6/20 0.46
F12 P00748 5/20 0.46
POLB P06746 1/20 0.46
KLK7 P49862 3/20 0.41
MAPT P10636 6/20 0.40
KMT2A Q03164 3/20 0.40
KLK5 Q9Y337 2/20 0.40
KLKB1 P03952 1/20 0.40
KLK1 P06870 1/20 0.40
KLK14 Q9P0G3 1/20 0.40
ST14 Q9Y5Y6 1/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
TP53 P04637 1/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
EGFR P00533 1/20 0.38
TUBB4A P04350 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2571839 0.81 KLK3 (0.66) KLK3F2F12KLK7MAPT
SCHEMBL14688829 0.79 F2 (0.55) F2POLBMAPTKMT2AKLKB1
SCHEMBL2567843 0.79 KLK3 (0.67) KLK3F2F12KLK7MAPT
SCHEMBL2568841 0.79 KLK3 (0.64) KLK3F2F12KLK7MAPT
SCHEMBL2552639 0.70 MAPT (0.78) F2POLBMAPTKMT2AKLKB1
SCHEMBL2689845 0.70 CYP2A6 (0.54) KLK3ALDH1A1CYP1A2CYP2C19
SCHEMBL2565569 0.69 F2 (0.48) KLK3F2F12MAPTKMT2A
SCHEMBL2568614 0.69 F2 (0.54) F2POLBMAPTKLKB1KLK1
SCHEMBL2551230 0.68 KLK3 (0.52) KLK3F2F12MAPTKMT2A
SCHEMBL30165671 0.67 CYP2A6 (0.50) POLBMAPTKMT2AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2560966-A2 MULTISUBSTITUTED AROMATIC COMPOUNDS AS INHIBITORS OF THROMBIN Verseon Corporation (US) 2013-02-27 EP disclosed
WO-2011126903-A2 MULTISUBSTITUTED AROMATIC COMPOUNDS AS INHIBITORS OF THROMBIN VERSEON, INC. (US) 2011-10-13 WO disclosed