SCHEMBL2568841

SCHEMBL2568841

CN(C)c1cccc(C(=O)n2nc(-c3cccnc3)cc2N)c1

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KLK3 P07288 7/20 0.64
ABL1 P00519 3/20 0.59
BCR P11274 3/20 0.59
TEK Q02763 1/20 0.49
ATR Q13535 1/20 0.47
HDAC1 Q13547 2/20 0.47
F12 P00748 3/20 0.46
FYN P06241 1/20 0.46
F2 P00734 1/20 0.44
MAPT P10636 1/20 0.44
KLK7 P49862 1/20 0.44
KMT2A Q03164 1/20 0.44
KLK14 Q9P0G3 1/20 0.44
KLK5 Q9Y337 1/20 0.44
ST14 Q9Y5Y6 1/20 0.44
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2571839 0.89 KLK3 (0.66) KLK3ABL1BCRHDAC1F12
SCHEMBL2567843 0.83 KLK3 (0.67) KLK3HDAC1F12F2MAPT
SCHEMBL14688962 0.79 MAPT (0.56) ABL1BCRTEKF2MAPT
SCHEMBL2561567 0.79 KLK3 (0.56) KLK3F12F2MAPTKLK7
SCHEMBL2562182 0.75 F2 (0.52) ABL1BCRTEKF2MAPT
SCHEMBL2551224 0.72 MAPT (0.78) F2MAPTKMT2ALMNA
SCHEMBL2551230 0.72 KLK3 (0.52) KLK3F12F2MAPTKMT2A
SCHEMBL2567005 0.70 F2 (0.58) F2MAPTKMT2ALMNA
SCHEMBL2689845 0.69 CYP2A6 (0.54) KLK3
SCHEMBL3791243 0.69 FYN (0.67) ABL1BCRATRFYNKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2560966-A2 MULTISUBSTITUTED AROMATIC COMPOUNDS AS INHIBITORS OF THROMBIN Verseon Corporation (US) 2013-02-27 EP disclosed
WO-2011126903-A2 MULTISUBSTITUTED AROMATIC COMPOUNDS AS INHIBITORS OF THROMBIN VERSEON, INC. (US) 2011-10-13 WO disclosed