SCHEMBL25623656

SCHEMBL25623656

NCCOc1ccc(OCC2CNCC[C@]2([SiH3])c2ccc(F)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.38
CYP19A1 P11511 1/20 0.38
ESR2 Q92731 1/20 0.38
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
LMNA P02545 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
SLC6A2 P23975 4/20 0.37
SLC6A4 P31645 4/20 0.37
SLC6A3 Q01959 3/20 0.37
HTR1A P08908 4/20 0.36
HTR2A P28223 4/20 0.36
DRD2 P14416 3/20 0.36
HRH1 P35367 3/20 0.36
DRD3 P35462 3/20 0.36
HTR2B P41595 3/20 0.36
HTR7 P34969 2/20 0.36
DRD1 P21728 1/20 0.36
DRD5 P21918 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25224507 0.69 GRK2 (0.65) ALDH1A1MEN1KMT2ALMNASLC6A2
SCHEMBL322907 0.68 TAAR1 (0.60) ESR1CYP19A1ESR2L3MBTL1DRD2
Hydrochloric Acid SCHEMBL25271410 0.68 GRK2 (0.67) ALDH1A1MEN1KMT2ALMNASLC6A2
Hydrochloric Acid SCHEMBL8865807 0.68 PLA2G7 (0.38) ALDH1A1HTR1AHTR2ADRD2HRH1
Hydrochloric Acid SCHEMBL321866 0.67 TAAR1 (0.58) ESR1CYP19A1ESR2ALDH1A1MEN1
SCHEMBL9633819 0.64 LTA4H (0.68) ESR1CYP19A1ESR2L3MBTL1LTA4H
SCHEMBL3163776 0.63 MAP2K1 (0.53) SLC6A2SLC6A4SLC6A3LTA4HTDP1
Hydrochloric Acid SCHEMBL1768943 0.62 MAP2K1 (0.52) SLC6A2SLC6A4SLC6A3LTA4HGRK2
SCHEMBL15645223 0.62 LTA4H (0.65) LTA4H
SCHEMBL15645221 0.62 LTA4H (0.65) LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023102477-A1 PERIPHERALLY AND LUMINALLY-RESTRICTED INHIBITORS OF THE SEROTONIN TRANSPORTER AS TREATMENTS FOR DISORDERS OF GASTROINTESTINAL MOTILITY THE JOHNS HOPKINS UNIVERSITY (US) 2023-06-08 WO disclosed