SCHEMBL2563418

SCHEMBL2563418

CCOC(=O)Oc1c(C)nn(-c2ccccc2)c1-c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.56
CYP2C19 P33261 3/20 0.56
CYP1A2 P05177 1/20 0.56
ALDH1A1 P00352 7/20 0.54
CYP3A4 P08684 2/20 0.54
PDE4D Q08499 1/20 0.52
HPGD P15428 2/20 0.47
NPSR1 Q6W5P4 4/20 0.47
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
KDM4E B2RXH2 3/20 0.46
KMT2A Q03164 2/20 0.44
GAA P10253 1/20 0.44
HSD17B10 Q99714 2/20 0.43
MAPT P10636 2/20 0.43
TP53 P04637 1/20 0.43
ALOX12 P18054 1/20 0.43
RAB9A P51151 1/20 0.43
MEN1 O00255 1/20 0.42
TSHR P16473 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2562342 0.89 ALDH1A1 (0.53) CYP2C9CYP2C19CYP1A2ALDH1A1CYP3A4
SCHEMBL2563146 0.88 ALDH1A1 (0.52) CYP2C9CYP2C19CYP1A2ALDH1A1CYP3A4
SCHEMBL2555825 0.85 PDE4D (0.63) ALDH1A1PDE4DHPGDNPSR1KDM4E
SCHEMBL2554340 0.80 KMT2A (0.56) CYP2C9CYP2C19ALDH1A1CYP3A4PDE4D
SCHEMBL12266478 0.79 PDE4D (0.73) CYP2C9CYP2C19CYP1A2ALDH1A1CYP3A4
SCHEMBL2919412 0.74 ALDH1A1 (0.73) CYP2C9CYP2C19CYP1A2ALDH1A1CYP3A4
SCHEMBL8422338 0.73 ALDH1A1 (0.68) CYP2C9CYP2C19CYP1A2ALDH1A1CYP3A4
SCHEMBL1997120 0.72 ALDH1A1 (0.53) CYP2C9CYP2C19CYP1A2ALDH1A1CYP3A4
SCHEMBL14132434 0.72 CYP2C9 (1.00) CYP2C9CYP2C19CYP1A2ALDH1A1CYP3A4
SCHEMBL12264387 0.72 ALDH1A1 (0.67) CYP2C9CYP2C19CYP1A2ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552895-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES Westfälische Wilhelms-Universität Münster (DE) 2013-02-06 EP disclosed
WO-2011120861-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES WESTFÄLISHE WILHELMS-UNIVERSITÄT MÜNSTER (DE) 2011-10-06 WO disclosed