SCHEMBL2554340

SCHEMBL2554340

CCOC(=O)Oc1c(-c2ccccc2)nn(-c2ccccc2)c1C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.56
MEN1 O00255 5/20 0.56
PDE4D Q08499 2/20 0.52
ALDH1A1 P00352 7/20 0.52
TSHR P16473 1/20 0.46
TP53 P04637 1/20 0.46
ALOX12 P18054 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
GAA P10253 1/20 0.44
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
NPSR1 Q6W5P4 2/20 0.43
MAPT P10636 1/20 0.43
RAB9A P51151 1/20 0.43
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2562342 0.89 ALDH1A1 (0.53) KMT2AMEN1PDE4DALDH1A1TSHR
SCHEMBL2553897 0.87 MEN1 (0.58) KMT2AMEN1PDE4DALDH1A1TSHR
SCHEMBL2555825 0.85 PDE4D (0.63) PDE4DALDH1A1TSHRTP53ALOX12
SCHEMBL2560207 0.84 MEN1 (0.40) KMT2AMEN1PDE4DALDH1A1CYP3A4
SCHEMBL2563418 0.80 CYP2C9 (0.56) KMT2AMEN1PDE4DALDH1A1TSHR
SCHEMBL2560863 0.79 ALDH1A1 (0.55) KMT2AMEN1ALDH1A1CYP3A4CYP2C9
SCHEMBL6264973 0.79 PDE4D (0.73) KMT2AMEN1PDE4DALDH1A1TP53
SCHEMBL2557760 0.78 MEN1 (0.48) KMT2AMEN1ALDH1A1TP53KDM4E
SCHEMBL2557580 0.78 KMT2A (0.48) KMT2AMEN1ALDH1A1TSHRTP53
SCHEMBL2563146 0.78 ALDH1A1 (0.52) KMT2APDE4DALDH1A1TSHRTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552895-B1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES Westfälische Wilhelms Universität Münster (DE) 2015-02-25 EP disclosed
EP-2552895-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES Westfälische Wilhelms-Universität Münster (DE) 2013-02-06 EP disclosed
WO-2011120861-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES WESTFÄLISHE WILHELMS-UNIVERSITÄT MÜNSTER (DE) 2011-10-06 WO disclosed