SCHEMBL2563804

SCHEMBL2563804

Nc1ncc(-c2ccc(N3CCNC(=O)C3)cc2)c(N)n1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DHFR P00374 10/20 0.46
ALOX5AP P20292 3/20 0.42
FEN1 P39748 2/20 0.42
GAK O14976 1/20 0.40
DPP4 P27487 1/20 0.39
AOC3 Q16853 1/20 0.39
PRKCH P24723 1/20 0.38
PRKCE Q02156 1/20 0.38
WNT3A P56704 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17907560 0.82 DHFR (0.56) DHFR
SCHEMBL30515653 0.82 DHFR (0.56) DHFR
SCHEMBL14694265 0.76 DHFR (0.58) DHFR
SCHEMBL2558872 0.75 DHFR (0.60) DHFR
SCHEMBL265154 0.74 DHFR (0.59) DHFR
SCHEMBL30560046 0.74 DHFR (0.59) DHFR
SCHEMBL3125646 0.74 DDB1 (0.46) GAKDPP4PRKCHPRKCE
SCHEMBL1991950 0.73 PIK3CA (0.50) ALOX5APFEN1GAKDPP4AOC3
SCHEMBL29660579 0.73 PIK3CA (0.50) ALOX5APFEN1GAKDPP4AOC3
SCHEMBL14320578 0.70 KDM4E (0.42) ALOX5APFEN1GAKAOC3PRKCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2558474-A1 2, 4-PYRIMIDINEDIAMINE COMPOUNDS AND PRODRUGS THEREOF AND THEIR USES Rigel Pharmaceuticals, Inc. (US) 2013-02-20 EP claimed
WO-2011130390-A1 2, 4-PYRIMIDINEDIAMINE COMPOUNDS AND PRODRUGS THEREOF AND THEIR USES RIGEL PHARMACEUTICALS, INC. (US) 2011-10-20 WO claimed