SCHEMBL30515653

SCHEMBL30515653

Nc1ncc(-c2ccc(N3CCNCC3)cc2)c(N)n1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DHFR P00374 7/20 0.56
TGFBR1 P36897 8/20 0.53
ACVR1 Q04771 9/20 0.49
HRH3 Q9Y5N1 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17907560 1.00 DHFR (0.56) DHFRTGFBR1ACVR1HRH3
SCHEMBL14694265 0.85 DHFR (0.58) DHFR
SCHEMBL2558872 0.84 DHFR (0.60) DHFR
SCHEMBL30560046 0.83 DHFR (0.59) DHFR
SCHEMBL265154 0.83 DHFR (0.59) DHFR
SCHEMBL2563804 0.82 DHFR (0.46) DHFR
SCHEMBL1199578 0.80 TGFBR1 (0.55) TGFBR1ACVR1
SCHEMBL14694244 0.78 DHFR (0.50) DHFR
SCHEMBL9167447 0.77 DHFR (0.59) DHFRHRH3
SCHEMBL30515507 0.75 FLT3 (0.45) TGFBR1ACVR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116514779-A 2, 4-disubstituted-5-fluoropyrimidine derivative and preparation method and application thereof 中南大学 2023-08-01 CN disclosed