SCHEMBL25643118

SCHEMBL25643118

COc1ccc(B2OC(C)(C)C(C)(C)O2)c2c(C#N)c(NC(=O)OC(C)(C)C)sc12

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 2/20 0.34
ALDH1A1 P00352 6/20 0.33
RXFP1 Q9HBX9 1/20 0.33
MAPT P10636 4/20 0.33
KDM4E B2RXH2 3/20 0.33
HPGD P15428 3/20 0.33
LMNA P02545 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
HSD17B10 Q99714 1/20 0.32
POLB P06746 1/20 0.32
NPC1 O15118 1/20 0.32
GAA P10253 1/20 0.31
MELK Q14680 1/20 0.31
ADORA2A P29274 1/20 0.31
PRMT5 O14744 1/20 0.31
WDR77 Q9BQA1 1/20 0.31
USP30 Q70CQ3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24757043 0.88 AAK1 (0.33) AAK1ALDH1A1MAPTKDM4EHPGD
SCHEMBL30537698 0.82 MEN1 (0.32) MEN1KMT2A
SCHEMBL25405428 0.82 MEN1 (0.32) MEN1KMT2A
SCHEMBL29813410 0.82 AAK1 (0.34) AAK1ALDH1A1RXFP1MAPTKDM4E
SCHEMBL23496728 0.82 AAK1 (0.34) AAK1ALDH1A1RXFP1MAPTKDM4E
SCHEMBL25643117 0.80 ALDH1A1 (0.38) AAK1ALDH1A1RXFP1MAPTKDM4E
SCHEMBL24717500 0.77 NPC1 (0.32) ALDH1A1MAPTKDM4EHPGDMEN1
SCHEMBL30014975 0.77 NPC1 (0.32) ALDH1A1MAPTKDM4EHPGDMEN1
SCHEMBL28807303 0.77 BRAF (0.30)
SCHEMBL29813229 0.77 BRAF (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023104018-A1 SUBSTITUTED BICYCLIC HETEROARYL COMPOUND AS KRAS G12D INHIBITOR 苏州浦合医药科技有限公司 2023-06-15 WO disclosed