SCHEMBL2564609

SCHEMBL2564609

Clc1ccc2c(c1)N1CCN(Cc3ccccc3)CC1CCN2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 1/20 0.47
DRD2 P14416 6/20 0.46
DRD4 P21917 3/20 0.46
DRD3 P35462 3/20 0.46
SIGMAR1 Q99720 3/20 0.44
CHRM3 P20309 3/20 0.42
CHRM2 P08172 2/20 0.42
BCHE P06276 2/20 0.41
ACHE P22303 2/20 0.41
BACE1 P56817 2/20 0.41
ALDH1A1 P00352 2/20 0.40
OPRM1 P35372 1/20 0.40
OPRK1 P41145 1/20 0.40
OPRL1 P41146 1/20 0.40
KDM4E B2RXH2 1/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1352182 0.88 DRD2 (0.51) DRD2DRD4DRD3SIGMAR1CHRM3
SCHEMBL691879 0.80 DRD2 (0.48) AVPR1ADRD2DRD4DRD3SIGMAR1
SCHEMBL2012961 0.78 CYP2D6 (0.47) DRD2DRD4DRD3SIGMAR1BCHE
SCHEMBL2017528 0.78 AVPR1A (0.42) AVPR1ADRD2DRD4ALDH1A1MAPT
SCHEMBL1350975 0.77 HTR3E (0.46) DRD2DRD4DRD3SIGMAR1CHRM3
SCHEMBL692590 0.76 CYP2D6 (0.44) DRD2DRD4DRD3SIGMAR1CHRM3
SCHEMBL2014482 0.76 CYP2D6 (0.44) DRD2DRD4DRD3SIGMAR1CHRM3
SCHEMBL692244 0.74 DRD2 (0.47) AVPR1ADRD2DRD4DRD3SIGMAR1
SCHEMBL691313 0.74 DRD2 (0.47) AVPR1ADRD2DRD4DRD3SIGMAR1
SCHEMBL2017936 0.74 HTR2C (0.60)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2560973-A1 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF Abbvie Inc. (US) 2013-02-27 EP claimed
WO-2011133182-A1 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF ABBOTT LABORATORIES (US) 2011-10-27 WO claimed