Bucloxic Acid

Bucloxic Acid

SCHEMBL25652

O=C(O)CCC(=O)c1ccc(C2CCCCC2)c(Cl)c1

nearest known ligand 0.59

Full drug profile on Sugi Atlas →

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 5/20 0.48
ALDH1A1 P00352 2/20 0.45
PTGDR Q13258 3/20 0.44
PTGER2 P43116 1/20 0.44
PKM P14618 1/20 0.43
TSHR P16473 1/20 0.43
S1PR1 P21453 2/20 0.43
USP5 P45974 3/20 0.41
KMT2A Q03164 1/20 0.41
THRB P10828 1/20 0.40
S1PR3 Q99500 1/20 0.40
HDAC6 Q9UBN7 2/20 0.40
NR4A2 P43354 1/20 0.40
CYP1A2 P05177 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bucloxic Acid SCHEMBL29473493 1.00 PTGDR2 (0.48) PTGDR2ALDH1A1PTGDRPTGER2PKM
SCHEMBL11013954 0.89 PTGDR2 (0.40) PTGDR2ALDH1A1PTGDRPTGER2
SCHEMBL12608946 0.88 KDM4E (0.44) PTGDR2ALDH1A1PTGDRPTGER2S1PR1
SCHEMBL11016878 0.86 PTGDR2 (0.38) PTGDR2ALDH1A1PTGDRPTGER2S1PR1
SCHEMBL13408604 0.86 HPGD (0.44) PTGDR2ALDH1A1PTGDRKMT2AHPGD
SCHEMBL28594167 0.84 ALDH1A1 (0.45) PTGDR2ALDH1A1PTGDRPTGER2THRB
SCHEMBL11016875 0.84 PTGDR2 (0.38) PTGDR2ALDH1A1PTGDRPTGER2THRB
SCHEMBL7317286 0.83 ALDH1A1 (0.45) PTGDR2ALDH1A1PTGDRPKMTSHR
SCHEMBL2760395 0.83 SIGMAR1 (0.43) PTGDR2ALDH1A1PTGDRPTGER2TSHR
SCHEMBL11015244 0.83 PTGDR2 (0.40) PTGDR2ALDH1A1PTGDRPTGER2THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 10800 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4470565-A1 METHOD FOR PREVENTING OR TREATING DISEASE OR DISORDER ASSOCIATED WITH ANTINEOPLASTIC AGENT OnQuality Pharmaceuticals China Ltd. (CN) 2024-12-04 EP claimed
US-RE50218-E1 Non-steroidal anti-inflammatory ophthalmic compositions SUN PHARMACEUTICAL INDUSTRIES LIMITED (IN) 2024-11-26 US claimed
CN-118742325-A Methods for preventing or treating diseases or conditions associated with antineoplastic agents 上海岸阔医药科技有限公司 2024-10-01 CN claimed
US-20240041935-A1 PREVENTION AND TREATMENT OF REPRODUCTIVE FAILURE BY REGENERATIVE CELLS AND ADJUVANTS CREATIVE MEDICAL TECHNOLOGIES, INC. (US) 2024-02-08 US claimed
EP-4308063-A1 PRE-FILLING SYSTEM TO ELIMINATE BUBBLES INSIDE CAPSULES HAVING A SOLID DOSAGE FORM Procaps SA (US) 2024-01-24 EP claimed
US-11771695-B2 Cannabinoid receptor modulators ARENA PHARMACEUTICALS, INC. (US) 2023-10-03 US claimed
WO-2023142996-A1 METHOD FOR PREVENTING OR TREATING DISEASE OR DISORDER ASSOCIATED WITH ANTINEOPLASTIC AGENT 上海岸阔医药科技有限公司 2023-08-03 WO claimed
EP-4185277-A1 SOFT SHELL GELATIN CAPSULES Procaps SA (US) 2023-05-31 EP claimed
US-20230088240-A1 ACCELERATING THE DRYING RATE OF SOFTGEL CAPSULES GLAS AMERICAS LLC 2023-03-23 US claimed
WO-2022197983-A1 PRE-FILLING SYSTEM TO ELIMINATE BUBBLES INSIDE CAPSULES HAVING A SOLID DOSAGE FORM PROCAPS SA (US) 2022-09-22 WO claimed
EP-0039051-B1 MANNICH-BASE HYDROXAMIC ACID PRODRUGS FOR THE IMPROVED BIOAVAILABILITY OF NON-STEROIDAL ANTI-INFLAMMATORY AGENTS, A PROCESS FOR PREPARING AND A PHARMACEUTICAL COMPOSITION CONTAINING THEM MERCK & CO. INC. (US) 1985-07-24 EP claimed
WO-1985002542-A1 ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING XANTHINES AND METHODS OF USING SAME SUNSHINE ABRAHAM 1985-06-20 WO claimed
US-4522826-A SYNERGISTIC MIXTURES RICHARDSON-VICKS INC. (US) 1985-06-11 US claimed
US-4486436-A Analgesic and anti-inflammatory compositions comprising caffeine and methods of using same ANALGESIC ASSOCIATES (US) 1984-12-04 US claimed
EP-0114886-A1 IMPROVED ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING CAFFEINE. SUNSHINE ABRAHAM (US) 1984-08-08 EP claimed
WO-1984000490-A1 IMPROVED ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING CAFFEINE AND METHODS OF USING SAME SUNSHINE ABRAHAM 1984-02-16 WO claimed
US-4376767-A ANTIBIOTICS AND PHARMACEUTICALS MERCK & CO., INC. (US) 1983-03-15 US claimed
EP-0055870-A1 Pyridylmethyl esters of selected bio-affecting carboxylic acids, process for preparing and pharmaceutical composition comprising the same MERCK & CO. INC. (US) 1982-07-14 EP claimed
EP-0051278-A1 Soft tertiary amine esters of bio-affecting carboxylic acids, processes for preparing and a pharmaceutical composition containing the same MERCK & CO. INC. (US) 1982-05-12 EP claimed
EP-0039051-A2 Mannich-base hydroxamic acid prodrugs for the improved bioavailability of non-steroidal anti-inflammatory agents, a process for preparing and a pharmaceutical composition containing them MERCK & CO. INC. (US) 1981-11-04 EP claimed