SCHEMBL256561

SCHEMBL256561

CC(=O)c1cc(C(=O)N2CCCC2c2ccccc2)cc(N(C)S(C)(=O)=O)c1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.46
HSP90AB1 P08238 1/20 0.46
RIPK1 Q13546 1/20 0.46
SCD5 Q86SK9 8/20 0.43
SCD O00767 5/20 0.43
ROCK2 O75116 2/20 0.43
PARP14 Q460N5 1/20 0.42
PARP10 Q53GL7 1/20 0.42
CCNC P24863 1/20 0.40
CDK8 P49336 1/20 0.40
TP53 P04637 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL167323 0.93 HSP90AA1 (0.47) HSP90AA1HSP90AB1RIPK1SCD5SCD
SCHEMBL164502 0.89 RIPK1 (0.46) HSP90AA1HSP90AB1RIPK1SCD5SCD
SCHEMBL256556 0.82 RIPK1 (0.53) HSP90AA1HSP90AB1RIPK1SCD5SCD
SCHEMBL166110 0.80 POLB (0.47) TP53HPGD
SCHEMBL175219 0.78 HSP90AA1 (0.47) HSP90AA1HSP90AB1RIPK1SCD5SCD
SCHEMBL167476 0.76 NPC1 (0.45) HSP90AA1HSP90AB1ROCK2
SCHEMBL8284954 0.74 BACE1 (0.66) SCD5SCDROCK2
SCHEMBL166963 0.74 RIPK1 (0.54) HSP90AA1HSP90AB1RIPK1SCD5SCD
SCHEMBL166455 0.73 CPT1A (0.38)
SCHEMBL715026 0.73 CPT1A (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012028563-A1 BACE INHIBITORS FOR USE IN THE TREATMENT OF DIABETES F. HOFFMANN-LA ROCHE AG (CH) 2012-03-08 WO disclosed