SCHEMBL256556

SCHEMBL256556

CC(=O)c1cc(C)cc(C(=O)N2CCCC2c2ccccc2)c1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.53
HSP90AA1 P07900 1/20 0.53
HSP90AB1 P08238 1/20 0.53
SCD5 Q86SK9 7/20 0.50
SCD O00767 4/20 0.50
ROCK2 O75116 2/20 0.48
CCNC P24863 1/20 0.48
CDK8 P49336 1/20 0.48
PARP14 Q460N5 1/20 0.47
PARP10 Q53GL7 1/20 0.47
PRMT5 O14744 2/20 0.45
WDR77 Q9BQA1 2/20 0.45
TACR1 P25103 1/20 0.45
TRPC3 Q13507 1/20 0.44
TRPC6 Q9Y210 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL166963 0.91 RIPK1 (0.54) RIPK1HSP90AA1HSP90AB1SCD5SCD
SCHEMBL168416 0.87 RIPK1 (0.53) RIPK1HSP90AA1HSP90AB1SCD5SCD
SCHEMBL256561 0.82 HSP90AA1 (0.46) RIPK1HSP90AA1HSP90AB1SCD5SCD
SCHEMBL10140476 0.82 NPC1 (0.57)
SCHEMBL164387 0.79 PARP14 (0.60) RIPK1HSP90AA1HSP90AB1SCD5SCD
SCHEMBL18143043 0.79 ROCK2 (0.57) RIPK1HSP90AA1HSP90AB1SCD5SCD
SCHEMBL6266657 0.78 TACR1 (0.47) RIPK1HSP90AA1HSP90AB1SCD5SCD
SCHEMBL8596155 0.77 PARP14 (0.62) RIPK1HSP90AA1HSP90AB1SCD5SCD
SCHEMBL31453129 0.77 SCD5 (0.58) RIPK1HSP90AA1HSP90AB1SCD5SCD
SCHEMBL166794 0.77 ROCK2 (0.60) RIPK1HSP90AA1HSP90AB1SCD5SCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012028563-A1 BACE INHIBITORS FOR USE IN THE TREATMENT OF DIABETES F. HOFFMANN-LA ROCHE AG (CH) 2012-03-08 WO disclosed