SCHEMBL2566491

SCHEMBL2566491

CCOC(=O)C(NC=C(C#N)C1CC1)C(=O)OCC

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.33
MAPT P10636 2/20 0.33
TSHR P16473 1/20 0.33
CYP2C9 P11712 1/20 0.33
NPSR1 Q6W5P4 2/20 0.32
KDM4E B2RXH2 1/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
RAB9A P51151 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
GAA P10253 2/20 0.30
POLB P06746 1/20 0.30
HIF1A Q16665 1/20 0.30
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2572768 0.78 CA12 (0.37) ALDH1A1MAPTTSHRCYP2C9NPSR1
SCHEMBL3004759 0.78 CYP1A2 (0.30)
SCHEMBL2572352 0.76 ALDH1A1 (0.38) ALDH1A1MAPTTSHRCYP2C9NPSR1
SCHEMBL11901718 0.71 CYP2C9 (0.38) ALDH1A1TSHRCYP2C9NPSR1KDM4E
SCHEMBL11901721 0.71 CYP2C9 (0.38) ALDH1A1TSHRCYP2C9NPSR1KDM4E
SCHEMBL13911904 0.71 CYP2C9 (0.38) ALDH1A1TSHRCYP2C9NPSR1KDM4E
SCHEMBL655921 0.67 RAB9A (0.44) ALDH1A1MAPTRAB9AGAAPOLB
SCHEMBL837941 0.66 MGAM (0.42) ALDH1A1MAPTCYP2C9NPSR1SMN1; SMN2
SCHEMBL12682934 0.65 CA12 (0.38) ALDH1A1CYP2C9NPSR1SMN1; SMN2L3MBTL1
SCHEMBL2825743 0.65 MEN1 (0.39) ALDH1A1MAPTTSHRRAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2382218-A1 DELTA-5-DESATURASE INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2011-11-02 EP disclosed