SCHEMBL2568293

SCHEMBL2568293

CN1CCc2ccc(NC(=O)[C@@H](CCCC(=O)O)NC(=O)Oc3ccc(Cl)s3)cc2CC1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 1/20 0.40
F10 P00742 6/20 0.36
ROCK2 O75116 1/20 0.35
SIRT5 Q9NXA8 4/20 0.35
SIRT1 Q96EB6 2/20 0.35
SIRT2 Q8IXJ6 2/20 0.35
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CA9 Q16790 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2566201 0.97 CCKBR (0.40) CCKBRF10ROCK2SIRT5SIRT1
SCHEMBL2567471 0.92 F10 (0.36) CCKBRF10ROCK2SIRT1SIRT2
SCHEMBL2572469 0.91 CCKBR (0.39) CCKBRF10ROCK2SIRT5SIRT1
SCHEMBL2572104 0.91 CCKBR (0.38) CCKBRF10ROCK2CA12CA1
SCHEMBL2572736 0.90 CCKBR (0.38) CCKBRF10ROCK2CA12CA1
SCHEMBL3382957 0.90 F10 (0.44) CCKBRF10ROCK2
SCHEMBL2567570 0.90 CCKBR (0.37) CCKBRF10ROCK2CA12CA1
SCHEMBL2566723 0.90 CCKBR (0.37) CCKBRF10ROCK2CA12CA1
SCHEMBL2573538 0.89 CCKBR (0.38) CCKBRF10ROCK2
SCHEMBL2574207 0.89 CCKBR (0.38) CCKBRF10ROCK2CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899330-B9 SUBSTITUTED GLYCINAMIDES HAVING AN ANTITHROMBOTIC AND FACTOR XA-INHIBITING EFFECT BOEHRINGER INGELHEIM INT (DE) 2011-11-09 EP disclosed
EP-1899330-B1 SUBSTITUTED GLYCINAMIDES HAVING AN ANTITHROMBOTIC AND FACTOR XA-INHIBITING EFFECT BOEHRINGER INGELHEIM INT (DE) 2010-11-24 EP disclosed