SCHEMBL256936

SCHEMBL256936

CCOc1ccc(-c2c(C)nn3c(-c4ccccc4)cc(N4CCC[C@H]4CO)nc23)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 10/20 0.48
MAPK1 P28482 4/20 0.48
THRB P10828 1/20 0.42
TP53 P04637 2/20 0.42
SYK P43405 1/20 0.40
BCL6 P41182 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.39
HSD17B10 Q99714 3/20 0.39
KDM4E B2RXH2 2/20 0.39
HPGD P15428 2/20 0.39
ALDH1A1 P00352 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 2/20 0.39
NPC1 O15118 1/20 0.39
LMNA P02545 1/20 0.38
FPR2 P25090 1/20 0.38
SCN9A Q15858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15020778 1.00 MAPT (0.48) MAPTMAPK1THRBTP53SYK
SCHEMBL15020622 0.92 FPR2 (0.47) MAPTMAPK1THRBHSD17B10KDM4E
SCHEMBL257541 0.91 MAPT (0.59) MAPTMAPK1TP53BCL6SMN1; SMN2
SCHEMBL15021012 0.91 MAPT (0.59) MAPTMAPK1TP53BCL6SMN1; SMN2
SCHEMBL15042196 0.91 MAPT (0.53) MAPTMAPK1TP53SYKBCL6
SCHEMBL15021014 0.90 MAPT (0.38) MAPTMAPK1THRBSYKBCL6
SCHEMBL15020749 0.89 MAPT (0.49) MAPTMAPK1TP53SYKBCL6
SCHEMBL15042156 0.89 MAPT (0.49) MAPTMAPK1TP53SYKBCL6
SCHEMBL15020597 0.89 FPR2 (0.40) MAPTMAPK1THRBHPGDFPR2
SCHEMBL15020600 0.89 FPR2 (0.40) MAPTMAPK1THRBHPGDFPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8975264-B2 Compound acting as a cannabinoid receptor-1 inhibitor AMOREPACIFIC CORPORATION (KR) 2015-03-10 US disclosed
US-8975264-B2 Compound acting as a cannabinoid receptor-1 inhibitor AMOREPACIFIC CORPORATION (KR) 2015-03-10 US disclosed
EP-2617723-A2 NOVEL COMPOUND ACTING AS A CANNABINOID RECEPTOR-1 INHIBITOR Amorepacific Corporation (KR) 2013-07-24 EP disclosed
US-20130158025-A1 NOVEL COMPOUND ACTING AS A CANNABINOID RECEPTOR-1 INHIBITOR AMOREPACIFIC CORPORATION (KR) 2013-06-20 US disclosed
US-20130158025-A1 NOVEL COMPOUND ACTING AS A CANNABINOID RECEPTOR-1 INHIBITOR AMOREPACIFIC CORPORATION (KR) 2013-06-20 US disclosed
WO-2012030170-A2 NOVEL COMPOUND ACTING AS A CANNABINOID RECEPTOR-1 INHIBITOR (주)아모레퍼시픽 (KR) 2012-03-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130158025-A1 NOVEL COMPOUND ACTING AS A CANNABINOID RECEPTOR-1 INHIBITOR CNR1, CNR2, GPR18 MAPT 2617/4885MAPK1 519/4885THRB 1690/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.