SCHEMBL2569466

SCHEMBL2569466

[Ir]c1cccc2ncc3ccccc3c12

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.57
GPR3 P46089 1/20 0.57
PDPK1 O15530 1/20 0.37
CYP1A2 P05177 3/20 0.37
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
MAPT P10636 2/20 0.35
LMNA P02545 1/20 0.35
RECQL P46063 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TOP2A P11388 2/20 0.35
ADORA3 P0DMS8 1/20 0.35
ALDH1A1 P00352 4/20 0.34
HPGD P15428 2/20 0.34
THRB P10828 1/20 0.34
HSD17B10 Q99714 1/20 0.34
EGFR P00533 1/20 0.34
HTT P42858 2/20 0.33
PDE10A Q9Y233 1/20 0.33
PDGFRB P09619 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30857515 0.81 KDM4E (0.61) KDM4EGPR3PDPK1CYP1A2NPC1
SCHEMBL9038627 0.79 KDM4E (0.59) KDM4EGPR3PDPK1CYP1A2NPC1
SCHEMBL27973182 0.79 GPR3 (0.64) KDM4EGPR3PDPK1CYP1A2NPC1
SCHEMBL10025808 0.78 GPR3 (0.68) KDM4EGPR3PDPK1CYP1A2NPC1
SCHEMBL23003529 0.78 KDM4E (0.57) KDM4EGPR3PDPK1CYP1A2NPC1
SCHEMBL460290 0.78 GPR3 (0.57) KDM4EGPR3PDPK1CYP1A2NPC1
SCHEMBL2422350 0.78 KDM4E (0.57) KDM4EGPR3PDPK1CYP1A2NPC1
SCHEMBL841678 0.78 KDM4E (0.57) KDM4EGPR3PDPK1CYP1A2NPC1
SCHEMBL329199 0.78 KDM4E (0.57) KDM4EGPR3PDPK1CYP1A2NPC1
SCHEMBL241588 0.78 KDM4E (0.57) KDM4EGPR3PDPK1CYP1A2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3081617-B1 BLUE EMITTER WITH HIGH EFFICIENCY BASED ON IMIDAZO [1,2-F] PHENANTHRIDINE IRIDIUM COMPLEXES UNIVERSAL DISPLAY CORP (US) 2017-11-15 EP disclosed
EP-3081617-A1 BLUE EMITTER WITH HIGH EFFICIENCY BASED ON IMIDAZO [1,2-F] PHENANTHRIDINE IRIDIUM COMPLEXES Universal Display Corporation (US) 2016-10-19 EP disclosed
EP-2382281-B1 BLUE EMITTER WITH HIGH EFFICIENCY BASED ON IMIDAZO [1,2-f] PHENANTHRIDINE IRIDIUM COMPLEXES UNIVERSAL DISPLAY CORP (US) 2016-04-27 EP disclosed
CN-103896991-A Blue emitter with high efficiency based on imidazo 1,2-f phenanthridine iridium complexes UNIVERSAL DISPLAY CORP 2014-07-02 CN disclosed
CN-102292409-A Blue emitters based on imidazo [1,2-f ] phenanthridine iridium complexes with high efficiency 2011-12-21 CN disclosed
EP-2382281-A1 BLUE EMITTER WITH HIGH EFFICIENCY BASED ON IMIDAZO [1,2-f]¨PHENANTHRIDINE IRIDIUM COMPLEXES Universal Display Corporation (US) 2011-11-02 EP disclosed
EP-2382281-A1 BLUE EMITTER WITH HIGH EFFICIENCY BASED ON IMIDAZO [1,2-f]¨PHENANTHRIDINE IRIDIUM COMPLEXES Universal Display Corporation (US) 2011-11-02 EP disclosed
WO-2010068876-A1 BLUE EMITTER WITH HIGH EFFICIENCY BASED ON IMIDAZO [1,2-f] PHENANTHRIDINE IRIDIUM COMPLEXES UNIVERSAL DISPLAY CORPORATION (US) 2010-06-17 WO disclosed
WO-2010068876-A1 BLUE EMITTER WITH HIGH EFFICIENCY BASED ON IMIDAZO [1,2-f] PHENANTHRIDINE IRIDIUM COMPLEXES UNIVERSAL DISPLAY CORPORATION (US) 2010-06-17 WO disclosed