SCHEMBL2570488

SCHEMBL2570488

CCc1cccc(CC)c1CCOc1ccc2[nH]nc(I)c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTK P33981 7/20 0.43
MAPK8 P45983 4/20 0.41
LMNA P02545 1/20 0.39
ATM Q13315 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HTR1A P08908 7/20 0.37
HTR1B P28222 7/20 0.37
HTR1D P28221 6/20 0.36
MTNR1A P48039 4/20 0.35
MTNR1B P49286 2/20 0.35
HSD17B10 Q99714 1/20 0.35
KDM4E B2RXH2 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C9 P11712 1/20 0.35
HTR2A P28223 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5953065 0.78 TTK (0.62) TTKMAPK8HSD17B10KDM4EMAPT
SCHEMBL2569461 0.77 TTK (0.74) TTKMAPK8CYP1A2CYP3A4CYP2D6
SCHEMBL2569442 0.76 TRPA1 (0.51) SMN1; SMN2KDM4E
SCHEMBL16023544 0.75 TTK (0.43) TTKMAPK8HTR1AHTR1BHTR1D
SCHEMBL2561086 0.75 TTK (0.59) TTKSMN1; SMN2HTR1ATP53CYP1A2
SCHEMBL2574384 0.70 TTK (0.55) TTKHTR1DKDM4EMAPT
SCHEMBL5952020 0.70 ALDH1A1 (0.53) TTKHSD17B10KDM4EMAPTHTR2A
SCHEMBL29923833 0.70 ALDH1A1 (0.53) TTKHSD17B10KDM4EMAPTHTR2A
SCHEMBL27688753 0.70 HTR1D (0.45) TTKMAPK8LMNAHTR1DKDM4E
SCHEMBL2558896 0.69 TRPA1 (0.49) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011123937-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2011-10-13 WO disclosed
WO-2011123937-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2011-10-13 WO disclosed