SCHEMBL257079

SCHEMBL257079

Cc1ccc(C#Cc2ccc(C(F)(F)F)cc2)o1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
KIF11 P52732 1/20 0.38
HTR1A P08908 1/20 0.35
HTR7 P34969 1/20 0.35
HTR6 P50406 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.34
EGFR P00533 1/20 0.34
PDGFRB P09619 1/20 0.34
KDR P35968 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
P2RY6 Q15077 1/20 0.33
GRM5 P41594 3/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PTPN1 P18031 1/20 0.32
PTPN6 P29350 1/20 0.32
PTPN11 Q06124 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9967692 0.80 KIF11 (0.36) KIF11PTGDR2P2RY6GRM5KDM4E
SCHEMBL14998069 0.77 KIF11 (0.56) KIF11P2RY6ALDH1A1EGLN1
SCHEMBL16747679 0.77 KIF11 (0.56) KIF11P2RY6ALDH1A1EGLN1
SCHEMBL10300065 0.75 KIF11 (0.47) KIF11PTGDR2GRM5ALDH1A1
SCHEMBL14997641 0.75 KIF11 (0.47) KIF11PTGDR2GRM5ALDH1A1
SCHEMBL10300108 0.75 KIF11 (0.47) KIF11PTGDR2GRM5ALDH1A1
SCHEMBL22779132 0.72 CYP2A6 (0.41) EGFRTDP1KDM4EALDH1A1LMNA
SCHEMBL20651264 0.70 TSHR (0.48) MAOAMAOBKIF11HTR1AHTR7
SCHEMBL3827578 0.69 KIF11 (0.48) MAOBKIF11ALDH1A1
SCHEMBL2830955 0.69 ALDH1A1 (0.59) KIF11GRM5ALDH1A1PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012028578-A1 SUBSTITUTED FUSED PYRIMIDINONES AND DIHYDROPYRIMIDINONES BAYER CROPSCIENCE AG (DE) 2012-03-08 WO disclosed