SCHEMBL2570852

SCHEMBL2570852

COC(=O)c1ccc2c(c1)CC(C)(C)C(c1cc(Cl)cc(Nc3ccccc3)c1)N2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 1/20 0.39
ALDH1A1 P00352 5/20 0.37
KMT2A Q03164 4/20 0.37
MEN1 O00255 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
HSD17B10 Q99714 1/20 0.34
MAPT P10636 4/20 0.33
RAB9A P51151 3/20 0.33
NPC1 O15118 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
GAPDH P04406 1/20 0.33
HSPA1A P0DMV8 1/20 0.33
PTPN7 P35236 1/20 0.33
ALOX5 P09917 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HTT P42858 1/20 0.33
AR P10275 1/20 0.33
ACHE P22303 1/20 0.33
CDC25A P30304 1/20 0.33
CDC25B P30305 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2574514 0.92 ALDH1A1 (0.36) ALDH1A1KMT2AMEN1HSD17B10MAPT
SCHEMBL2530592 0.89 RAB9A (0.43) ALDH1A1KMT2AMEN1SMN1; SMN2HSD17B10
SCHEMBL2575481 0.88 CRBN (0.45) CRBNALDH1A1KMT2AMEN1SMN1; SMN2
SCHEMBL2535656 0.84 ALDH1A1 (0.40) CRBNALDH1A1KMT2AMEN1SMN1; SMN2
SCHEMBL2527478 0.81 MEN1 (0.39) ALDH1A1KMT2AMEN1SMN1; SMN2MAPT
SCHEMBL2530178 0.80 NPC1 (0.40) ALDH1A1KMT2AMEN1RAB9ANPC1
SCHEMBL2531679 0.80 ALDH1A1 (0.39) ALDH1A1KMT2AMEN1SMN1; SMN2HSD17B10
SCHEMBL2574768 0.79 MAPT (0.40) CRBNALDH1A1KMT2AMEN1SMN1; SMN2
SCHEMBL2533556 0.78 ALDH1A1 (0.41) ALDH1A1KMT2AMEN1SMN1; SMN2MAPT
SCHEMBL2535710 0.78 PTPN1 (0.49) ALDH1A1KMT2AMEN1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2558449-A1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2013-02-20 EP disclosed
WO-2011128251-A1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2011-10-20 WO disclosed