SCHEMBL2570965

SCHEMBL2570965

COc1ccc(C2(O)c3ccc(O)c(C)c3OCC2c2ccc(OC)c(OC)c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 3/20 0.40
ALOX12 P18054 3/20 0.40
ALOX5 P09917 1/20 0.36
PTPN1 P18031 1/20 0.36
PPARG P37231 1/20 0.36
PPARD Q03181 1/20 0.36
LMNA P02545 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
ALDH1A1 P00352 2/20 0.35
GAA P10253 1/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
MAPK10 P53779 1/20 0.35
BACE1 P56817 1/20 0.35
CYP3A4 P08684 2/20 0.34
CYP19A1 P11511 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13673338 0.91 SMN1; SMN2 (0.38) ALOX15ALOX12LMNAKDM4EMAPT
SCHEMBL2569873 0.91 ALOX15 (0.42) ALOX15ALOX12ALOX5PTPN1KDM4E
SCHEMBL2563485 0.91 ALOX15 (0.46) ALOX15ALOX12KDM4EMAPTALDH1A1
SCHEMBL2563436 0.90 ALOX15 (0.40) ALOX15ALOX12ALOX5PTPN1PPARG
SCHEMBL13673358 0.89 ALOX15 (0.41) ALOX15ALOX12LMNAGAABACE1
SCHEMBL2570309 0.88 ALOX15 (0.43) ALOX15ALOX12MAPTALDH1A1GAA
SCHEMBL2566790 0.87 ALOX15 (0.39) ALOX15ALOX12LMNAKDM4EMAPT
SCHEMBL2568306 0.86 ALOX15 (0.38) ALOX15ALOX12LMNAKDM4EMAPT
SCHEMBL2568812 0.86 ALOX15 (0.38) ALOX15ALOX12LMNAKDM4EMAPT
SCHEMBL12063383 0.85 ALDH1A1 (0.33) ALOX15ALOX12LMNAKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1794141-B1 SUBSTITUTED CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY MARSHALL EDWARDS INC (US) 2011-11-09 EP claimed
US-20160287555-A1 SUBSTITUTED CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RESEARCH PTY LTD (AU) 2016-10-06 US disclosed
US-20160287555-A1 SUBSTITUTED CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RESEARCH PTY LTD (AU) 2016-10-06 US disclosed
US-9381186-B2 Substituted chroman derivatives, medicaments and use in therapy MEI PHARMA, INC. (US) 2016-07-05 US disclosed
US-9381186-B2 Substituted chroman derivatives, medicaments and use in therapy MEI PHARMA, INC. (US) 2016-07-05 US disclosed
US-20150352074-A1 SUBSTITUTED CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RESEARCH PTY LTD (AU) 2015-12-10 US disclosed
US-20150352074-A1 SUBSTITUTED CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RESEARCH PTY LTD (AU) 2015-12-10 US disclosed
US-9138478-B2 Substituted chroman derivatives, medicaments and use in therapy MEI PHARMA, INC. (US) 2015-09-22 US disclosed
US-9138478-B2 Substituted chroman derivatives, medicaments and use in therapy MEI PHARMA, INC. (US) 2015-09-22 US disclosed
EP-2407462-B1 Substituted chroman derivatives, medicaments and use in therapy MARSHALL EDWARDS INC (US) 2014-07-30 EP disclosed
US-20140170243-A1 SUBSTITUTED CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY MEI PHARMA, INC. (US) 2014-06-19 US disclosed
US-20140170243-A1 SUBSTITUTED CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY MEI PHARMA, INC. (US) 2014-06-19 US disclosed
US-20120114766-A1 SUBSTITUTED CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY MARSHALL EDWARDS, INC. (US) 2012-05-10 US disclosed
US-20120114766-A1 SUBSTITUTED CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY MARSHALL EDWARDS, INC. (US) 2012-05-10 US disclosed
US-8084628-B2 Substituted chroman derivatives, medicaments and use in therapy MARSHALL EDWARDS, INC. (US) 2011-12-27 US disclosed
US-8084628-B2 Substituted chroman derivatives, medicaments and use in therapy MARSHALL EDWARDS, INC. (US) 2011-12-27 US disclosed
US-20090317490-A1 SUBSTITUTED CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RESEARCH PTY LTD. (AU) 2009-12-24 US disclosed
US-20090317490-A1 SUBSTITUTED CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RESEARCH PTY LTD. (AU) 2009-12-24 US disclosed
US-7601855-B2 anticancer agents; chemotherapeutic selective agents NOVOGEN RESEARCH PTY LTD (AU) 2009-10-13 US disclosed
US-7601855-B2 anticancer agents; chemotherapeutic selective agents NOVOGEN RESEARCH PTY LTD (AU) 2009-10-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150352074-A1 SUBSTITUTED CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY CDYL, XPA, TP53 ALOX15 4170/4885ALOX12 4177/4885ALOX5 3004/4885
US-20140170243-A1 SUBSTITUTED CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY CDYL, XPA, TP53 ALOX15 4170/4885ALOX12 4177/4885ALOX5 3004/4885
US-20120114766-A1 SUBSTITUTED CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY CDYL, XPA, TP53 ALOX15 4170/4885ALOX12 4177/4885ALOX5 3004/4885
US-20090317490-A1 SUBSTITUTED CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY CDYL, XPA, TP53 ALOX15 4170/4885ALOX12 4177/4885ALOX5 3004/4885
US-20160287555-A1 SUBSTITUTED CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY CDYL, XPA, TP53 ALOX15 4170/4885ALOX12 4177/4885ALOX5 3004/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.