SCHEMBL25720301

SCHEMBL25720301

CCOc1cccc(-c2n[nH]cc2-c2ccncc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 3/20 0.52
TTK P33981 3/20 0.47
MAPK14 Q16539 2/20 0.46
BRAF P15056 1/20 0.46
NTRK1 P04629 1/20 0.46
FGFR2 P21802 2/20 0.44
FGFR3 P22607 2/20 0.44
GAA P10253 2/20 0.43
MAPT P10636 2/20 0.43
KDM4E B2RXH2 1/20 0.43
THRB P10828 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
MAPK13 O15264 1/20 0.43
RAF1 P04049 1/20 0.43
MAPK12 P53778 1/20 0.43
MAPK11 Q15759 1/20 0.43
EGFR P00533 1/20 0.42
FGFR1 P11362 1/20 0.42
ROCK2 O75116 1/20 0.42
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17088191 0.83 ALDH1A1 (0.52) TTKMAPTKDM4ETDP1CYP3A4
SCHEMBL25720323 0.83 FGFR2 (0.44) S1PR1TTKFGFR2FGFR3GAA
SCHEMBL25418869 0.82 EGFR (0.43) TTKMAPK14BRAFNTRK1FGFR2
SCHEMBL31481576 0.82 EGFR (0.43) TTKMAPK14BRAFNTRK1FGFR2
SCHEMBL31481543 0.81 EGFR (0.50) S1PR1MAPK14BRAFNTRK1FGFR2
SCHEMBL25419956 0.81 MEN1 (0.51) MAPTKDM4ETHRBTDP1EGFR
SCHEMBL31481571 0.81 MEN1 (0.51) MAPTKDM4ETHRBTDP1EGFR
SCHEMBL25418273 0.81 EGFR (0.50) S1PR1MAPK14BRAFNTRK1FGFR2
SCHEMBL5496607 0.78 GRM4 (0.51) TTKMAPK14NTRK1FGFR2FGFR3
SCHEMBL25199043 0.78 CYP11B1 (0.54) EGFRROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023091873-A1 GRAM-NEGATIVE SPECIFIC ANTIBIOTICS SPARING EFFECT ON GUT MICROBIOME THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2023-05-25 WO disclosed