SCHEMBL2574254

SCHEMBL2574254

Cc1cnn2c(Cl)c3c(nc12)CCN(C(=O)O)CC3

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.36
TSHR P16473 4/20 0.36
ALDH1A1 P00352 5/20 0.35
HSD17B10 Q99714 4/20 0.35
KDM4E B2RXH2 4/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C19 P33261 2/20 0.35
KMT2A Q03164 2/20 0.33
MAPK1 P28482 2/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
HCRTR1 O43613 1/20 0.32
GAA P10253 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
SPR P35270 2/20 0.31
P2RX7 Q99572 1/20 0.31
HSP90AA1 P07900 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9948087 0.84 SPR (0.44) TSHRKMT2AMEN1MAPTSPR
SCHEMBL10217549 0.75 HTR2C (0.41) HPGDTSHRALDH1A1HSD17B10KDM4E
SCHEMBL2565601 0.74 HTR2C (0.44) P2RX7PDE10A
SCHEMBL9948065 0.71 SPR (0.40) HPGDHSD17B10KMT2AMEN1MAPT
SCHEMBL10217519 0.71 SPR (0.39) ALDH1A1KMT2AMEN1MAPTGAA
SCHEMBL10217543 0.71 SPR (0.45) MAPTSPR
SCHEMBL10217544 0.68 SPR (0.44) TSHRKMT2AMEN1MAPTSPR
SCHEMBL2570616 0.68 HTR2C (0.40) HPGDTSHRALDH1A1HSD17B10KDM4E
SCHEMBL28830137 0.67 CHRM4 (0.39) ALDH1A1CYP1A2MAPK1HSP90AA1HSP90AB1
SCHEMBL28894031 0.66 C5AR1 (0.32) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2384328-A1 6,7,8,9-TETRAHYDRO-5H-1,4,7,10A-TETRAAZA-CYCLOHEPT[F]INDENE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESS FOR PREPARING THEM Boehringer Ingelheim International GmbH (DE) 2011-11-09 EP disclosed
WO-2010060952-A1 6,7,8,9-TETRAHYDRO-5H-1,4,7,10A-TETRAAZA-CYCLOHEPT[F]INDENE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-06-03 WO disclosed