SCHEMBL25746271

SCHEMBL25746271

COc1ccc2c(S)nc(C)nc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.47
MPO P05164 1/20 0.46
KDM4E B2RXH2 7/20 0.44
ALDH1A1 P00352 6/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
POLB P06746 2/20 0.44
LMNA P02545 2/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
NQO2 P16083 1/20 0.44
RAB9A P51151 1/20 0.44
KMT2A Q03164 1/20 0.44
APP P05067 2/20 0.43
HPGD P15428 3/20 0.43
HSD17B10 Q99714 2/20 0.43
TSHR P16473 1/20 0.43
HBB P68871 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31391492 1.00 NPSR1 (0.47) NPSR1MPOKDM4EALDH1A1SMN1; SMN2
SCHEMBL25284840 0.86 POLB (0.54) KDM4EALDH1A1SMN1; SMN2POLBLMNA
SCHEMBL30466795 0.86 POLB (0.54) KDM4EALDH1A1SMN1; SMN2POLBLMNA
SCHEMBL9283331 0.82 NPSR1 (0.60) NPSR1MPOKDM4EALDH1A1SMN1; SMN2
SCHEMBL8145986 0.81 NPSR1 (0.48) NPSR1MPOKDM4EALDH1A1SMN1; SMN2
SCHEMBL857219 0.79 KDM4E (0.49) NPSR1MPOKDM4EALDH1A1SMN1; SMN2
SCHEMBL20813453 0.79 APP (0.48) NPSR1MPOKDM4EALDH1A1SMN1; SMN2
SCHEMBL30640287 0.79 KDM4E (0.49) NPSR1MPOKDM4EALDH1A1SMN1; SMN2
SCHEMBL14819968 0.79 DHFR (0.52) NPSR1MPOKDM4EALDH1A1SMN1; SMN2
SCHEMBL31391484 0.78 CYP1A2 (0.41) KDM4EALDH1A1LMNANQO2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023118507-A2 COMPOUNDS AND USE THEREOF AS HDAC6 INHIBITORS AUGUSTINE THERAPEUTICS (BE) 2023-06-29 WO disclosed