SCHEMBL8145986

SCHEMBL8145986

COc1ccc2c(OC)nc(C)nc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.48
MPO P05164 1/20 0.47
ACHE P22303 1/20 0.47
KDM4E B2RXH2 5/20 0.46
ALDH1A1 P00352 5/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
LMNA P02545 2/20 0.46
POLB P06746 2/20 0.46
MEN1 O00255 1/20 0.46
NPC1 O15118 1/20 0.46
NQO2 P16083 1/20 0.46
RAB9A P51151 1/20 0.46
KMT2A Q03164 1/20 0.46
HTT P42858 1/20 0.45
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 1/20 0.44
VDR P11473 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2B6 P20813 1/20 0.44
AHR P35869 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8131948 0.86 KDM4E (0.51) KDM4EALDH1A1SMN1; SMN2LMNAPOLB
SCHEMBL9283331 0.84 NPSR1 (0.60) NPSR1MPOACHEKDM4EALDH1A1
SCHEMBL8149547 0.82 ACHE (0.47) NPSR1MPOACHEKDM4EALDH1A1
SCHEMBL25746271 0.81 NPSR1 (0.47) NPSR1MPOACHEKDM4EALDH1A1
SCHEMBL20813453 0.81 APP (0.48) NPSR1MPOACHEKDM4EALDH1A1
SCHEMBL31391492 0.81 NPSR1 (0.47) NPSR1MPOACHEKDM4EALDH1A1
SCHEMBL14819968 0.81 DHFR (0.52) NPSR1MPOACHEKDM4EALDH1A1
SCHEMBL857219 0.81 KDM4E (0.49) NPSR1MPOACHEKDM4EALDH1A1
SCHEMBL30640287 0.81 KDM4E (0.49) NPSR1MPOACHEKDM4EALDH1A1
SCHEMBL24392233 0.78 NPSR1 (0.44) NPSR1MPOACHEKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009005677-A2 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2009-01-08 WO disclosed