SCHEMBL25752263

SCHEMBL25752263

CCN(C(=O)NC)c1cccnc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.55
CYP2C19 P33261 2/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2B6 P20813 1/20 0.50
KDM4E B2RXH2 2/20 0.48
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
NPSR1 Q6W5P4 3/20 0.45
MAPT P10636 2/20 0.45
GFER P55789 2/20 0.45
ALDH1A1 P00352 5/20 0.43
LMNA P02545 2/20 0.43
TSHR P16473 2/20 0.42
GLA P06280 1/20 0.42
TRPV1 Q8NER1 1/20 0.41
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
GAA P10253 2/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19305858 0.88 HTT (0.55) HTTCYP2C19CYP3A4CYP2C9CYP2B6
SCHEMBL6671752 0.83 HTT (0.65) HTTCYP2C19CYP3A4CYP2C9CYP2B6
SCHEMBL28060973 0.82 MEN1 (0.73) HTTCYP2C19CYP3A4CYP2C9CYP2B6
SCHEMBL14539624 0.82 HTT (0.59) HTTCYP2C19CYP3A4CYP2C9CYP2B6
SCHEMBL27624091 0.81 HTT (0.57) HTTCYP2C19CYP3A4CYP2C9CYP2B6
SCHEMBL666963 0.81 HTT (0.57) HTTCYP2C19CYP3A4CYP2C9CYP2B6
SCHEMBL966694 0.80 MEN1 (0.69) HTTCYP2C19CYP3A4CYP2C9MEN1
SCHEMBL2485280 0.78 MKNK1 (0.43) HTTCYP3A4NPSR1MAPTGFER
SCHEMBL4670467 0.77 HTT (0.54) HTTCYP2C19CYP3A4CYP2C9CYP2B6
SCHEMBL12978259 0.75 HTT (0.66) HTTCYP2C19CYP3A4CYP2C9CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023116390-A1 PYRIMIDINE-2(1H)-ONE-FUSED BICYCLIC COMPOUND HAVING MAT2A INHIBITORY ACTIVITY AND USE THEREOF 上海海和药物研究开发股份有限公司 2023-06-29 WO disclosed