SCHEMBL25757650

SCHEMBL25757650

O=C1NCc2c1ccc1ocnc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 3/20 0.40
CLK4 Q9HAZ1 3/20 0.40
CDK5 Q00535 2/20 0.40
PIM1 P11309 2/20 0.40
ROCK1 Q13464 2/20 0.40
CSNK1A1 P48729 1/20 0.40
LRRK2 Q5S007 1/20 0.40
DYRK1B Q9Y463 1/20 0.40
LTK P29376 1/20 0.36
MST1R Q04912 1/20 0.36
KDR P35968 2/20 0.33
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
CYP17A1 P05093 1/20 0.33
CYP3A4 P08684 1/20 0.33
MAP4K1 Q92918 1/20 0.33
PLK4 O00444 1/20 0.33
ROCK2 O75116 1/20 0.33
MAP4K4 O95819 1/20 0.33
PRKCG P05129 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16335317 0.74 DYRK1A (0.40) DYRK1ACLK4CDK5PIM1ROCK1
SCHEMBL16535812 0.69 LMNA (0.53) DYRK1ACLK4CDK5PIM1ROCK1
SCHEMBL28730418 0.68 NOTUM (0.42)
SCHEMBL25757654 0.68 CLK4 (0.42) DYRK1ACLK4CDK5PIM1ROCK1
SCHEMBL10054248 0.67 HTR2A (0.39) DYRK1A
SCHEMBL24466337 0.63 CDK5 (0.46) DYRK1ACLK4CDK5PIM1ROCK1
SCHEMBL31264207 0.63 CDK5 (0.46) DYRK1ACLK4CDK5PIM1ROCK1
SCHEMBL15566157 0.63 CLK4 (0.46) DYRK1ACLK4CDK5PIM1ROCK1
SCHEMBL16921409 0.63 CDK5 (0.46) DYRK1ACLK4CDK5PIM1ROCK1
SCHEMBL30842095 0.63 CDK5 (0.46) DYRK1ACLK4CDK5PIM1ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023098880-A1 FUSED RING DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 上海翰森生物医药科技有限公司 2023-06-08 WO disclosed