SCHEMBL25757925

SCHEMBL25757925

O=C(NI)c1cc(F)cc(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.47
GAA P10253 1/20 0.46
HDAC3 O15379 2/20 0.43
HDAC6 Q9UBN7 2/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
DDR1 Q08345 1/20 0.43
VNN1 O95497 3/20 0.43
HDAC8 Q9BY41 1/20 0.43
TACR1 P25103 1/20 0.41
P2RX1 P51575 2/20 0.41
RHOC P08134 1/20 0.40
RHOA P61586 1/20 0.40
NOTUM Q6P988 1/20 0.39
CSF1R P07333 1/20 0.39
AURKA O14965 1/20 0.39
ENPP2 Q13822 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14214023 0.82 CES2 (0.47) CES2GAAHDAC3HDAC6HDAC1
SCHEMBL30554615 0.79 P2RX1 (0.65) HDAC3HDAC6HDAC8P2RX1RHOC
SCHEMBL3246188 0.79 P2RX1 (0.65) HDAC3HDAC6HDAC8P2RX1RHOC
SCHEMBL13753158 0.79 DDR1 (0.47) CES2GAAHDAC3HDAC6HDAC1
SCHEMBL27757817 0.79 CES2 (0.56) CES2GAAHDAC3HDAC6HDAC1
SCHEMBL13753151 0.78 NPSR1 (0.63) CES2GAADDR1HDAC8NOTUM
SCHEMBL13753001 0.78 DDR1 (0.55) CES2GAADDR1VNN1TACR1
SCHEMBL586089 0.77 HCAR1 (0.55) CES2VNN1
SCHEMBL1827001 0.77 CES2 (0.54) CES2GAAHDAC3HDAC6HDAC1
SCHEMBL30770849 0.77 HCAR1 (0.55) CES2VNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023168378-A1 PI3KA INHIBITORS SYNNOVATION THERAPEUTICS, INC. (US) 2023-09-07 WO disclosed
WO-2023098880-A1 FUSED RING DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 上海翰森生物医药科技有限公司 2023-06-08 WO disclosed