SCHEMBL257599

SCHEMBL257599

Cc1ccc(COCc2cccc3ccccc23)cc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.50
TACR1 P25103 1/20 0.50
HSP90AB1 P08238 1/20 0.44
CYP1A2 P05177 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP2D6 P10635 1/20 0.43
LMNA P02545 1/20 0.43
PKM P14618 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
AKR1B1 P15121 2/20 0.43
FFAR1 O14842 1/20 0.43
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.41
DHODH Q02127 1/20 0.40
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707213 0.86 TSHR (0.58) TACR1HSP90AB1CYP1A2CYP2C19CYP2D6
SCHEMBL31012122 0.84 CYP1A2 (0.56) HSP90AB1CYP1A2CYP2C19CYP2D6CYP2C9
SCHEMBL4850585 0.84 CYP1A2 (0.56) HSP90AB1CYP1A2CYP2C19CYP2D6CYP2C9
SCHEMBL31065555 0.83 IDO1 (0.46) TACR1HSP90AB1CYP1A2CYP2C19LMNA
SCHEMBL10269557 0.80 FFAR1 (0.43) HSP90AB1L3MBTL1AKR1B1FFAR1
SCHEMBL29417924 0.79 CYP2C19 (0.53) CYP1A2CYP2C19CYP2D6CYP2C9
SCHEMBL7629984 0.79 CYP2C19 (0.53) CYP1A2CYP2C19CYP2D6CYP2C9
SCHEMBL12270341 0.79 KCNH2 (0.51) KCNH2TACR1TSHRDHODH
Hydroxyamine SCHEMBL8924246 0.78 MEN1 (0.53) HSP90AB1CYP1A2CYP2C19CYP2D6CYP2C9
SCHEMBL15249121 0.78 PARP10 (0.61) KCNH2LMNAAKR1B1FFAR1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2399585-A1 Boronic acids and esters as inhibitors of fatty acid amide hydrolase Infinity Pharmaceuticals, Inc. (US) 2011-12-28 EP disclosed
EP-2073816-B1 BORONIC ACIDS AND ESTERS AS INHIBITORS OF FATTY ACID AMIDE HYDROLASE INFINITY PHARMACEUTICALS INC (US) 2011-09-14 EP disclosed